SCHEMBL8620404

SCHEMBL8620404

COc1ccc(C(C)C)cc1CNCC(NC1CCCC1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.50
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
TACR1 P25103 5/20 0.42
CFTR P13569 1/20 0.42
GAA P10253 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
LMNA P02545 1/20 0.41
SGPL1 O95470 1/20 0.40
BCHE P06276 1/20 0.39
PDE4A P27815 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6555183 0.99 CYP2D6 (0.49) CYP2D6MEN1KMT2ATACR1CFTR
SCHEMBL6555294 0.87 MEN1 (0.61) MEN1KMT2ATACR1L3MBTL1LMNA
SCHEMBL6556099 0.85 MEN1 (0.60) MEN1KMT2ATACR1L3MBTL1LMNA
SCHEMBL6556931 0.85 MEN1 (0.60) MEN1KMT2ATACR1L3MBTL1LMNA
SCHEMBL8621981 0.85 TACR1 (0.48) CYP2D6MEN1KMT2ATACR1CFTR
SCHEMBL8620048 0.85 SGPL1 (0.49) MEN1KMT2AGAAL3MBTL1SGPL1
SCHEMBL7713389 0.85 TACR1 (0.48) CYP2D6MEN1KMT2ATACR1CFTR
Hydrochloric Acid SCHEMBL8620287 0.84 MEN1 (0.59) MEN1KMT2ATACR1L3MBTL1LMNA
SCHEMBL6555248 0.84 MEN1 (0.61) MEN1KMT2ATACR1L3MBTL1LMNA
SCHEMBL6556838 0.84 SGPL1 (0.48) MEN1KMT2AGAAL3MBTL1SGPL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0613458-B1 ACYCLIC ETHYLENEDIAMINE DERIVATIVES AS SUBSTANCE P RECEPTOR ANTAGONISTS PFIZER (US) 1998-01-07 EP disclosed
US-5521220-A Acyclic ethylenediamine derivatives PFIZER INC. (US) 1996-05-28 US disclosed
WO-1993010073-A1 ACYCLIC ETHYLENEDIAMINE DERIVATIVES AS SUBSTANCE P RECEPTOR ANTAGONISTS PFIZER INC. (US) 1993-05-27 WO disclosed