SCHEMBL8620773

SCHEMBL8620773

CC(C)C(Cl)(C(=O)O)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.55
CYP2D6 P10635 2/20 0.55
HIF1A Q16665 2/20 0.44
CYP2C19 P33261 1/20 0.44
TSHR P16473 2/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
KIF11 P52732 1/20 0.40
KCNN4 O15554 1/20 0.39
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1669593 0.84 CYP1A2 (0.52) CYP1A2CYP2D6HIF1ACYP2C19TSHR
SCHEMBL28342296 0.81 CYP1A2 (0.56) CYP1A2CYP2D6HIF1ACYP2C19TSHR
SCHEMBL11839409 0.77 PIN1 (0.47) CYP1A2CYP2D6TSHRMAPTKMT2A
SCHEMBL27812340 0.76 CYP1A2 (0.40) CYP1A2CYP2D6HIF1ACYP2C19MAPT
SCHEMBL13641402 0.74 CYP2D6 (0.59) CYP1A2CYP2D6HIF1ACYP2C19TSHR
SCHEMBL9435860 0.73 CYP1A2 (0.47) CYP1A2CYP2D6HIF1ACYP2C19TSHR
SCHEMBL21268837 0.72 CYP2D6 (0.57) CYP1A2CYP2D6HIF1ACYP2C19TSHR
SCHEMBL28875699 0.72 CYP2D6 (0.57) CYP1A2CYP2D6HIF1ACYP2C19TSHR
SCHEMBL21269485 0.72 CYP2D6 (0.57) CYP1A2CYP2D6HIF1ACYP2C19TSHR
SCHEMBL21269904 0.72 CYP2D6 (0.57) CYP1A2CYP2D6HIF1ACYP2C19TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5786428-A POLYMER MATRIX OF UNSATURATED MONOMER AND METAL COMPLEX HAVING A LIGAND AND A POLYMERIZABLE UNSATURATED MOIETY; EFFICIENT, RAPID AND SIMPLE PURIFICATION; MEDICAL DIAGNOSIS; CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 1998-07-28 US claimed
EP-0114012-B1 ESTERS OF CYCLOPROPANE-CARBOXYLIC ACIDS AND UNSATURATED ALIPHATIC ALCOHOLS, PROCESS AND INTERMEDIATES OF PREPARATION AND PESTICIDAL COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1986-10-08 EP claimed
CN-104114020-A Plant growing system and method employing said system OMS INVESTMENTS INC 2014-10-22 CN disclosed
CN-101500410-A Granular controlled release agrochemical compositions and process for preparing same OMS INVEST INC (US) 2009-08-05 CN disclosed
US-5786428-A POLYMER MATRIX OF UNSATURATED MONOMER AND METAL COMPLEX HAVING A LIGAND AND A POLYMERIZABLE UNSATURATED MOIETY; EFFICIENT, RAPID AND SIMPLE PURIFICATION; MEDICAL DIAGNOSIS; CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 1998-07-28 US disclosed
EP-0339599-A2 Process for producing acylaromatic compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1989-11-02 EP disclosed