SCHEMBL8622935

SCHEMBL8622935

CC[C@](Cc1ccccc1)(NC(=O)[C@H](CC(N)=O)NC(=O)c1ccc2ccccc2n1)N(CCC(C)C)S(=O)(=O)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 3/20 0.45
CYP3A4 P08684 3/20 0.44
LMNA P02545 2/20 0.44
USP2 O75604 1/20 0.44
CYP2D6 P10635 1/20 0.44
ALDH1A1 P00352 1/20 0.44
TP53 P04637 1/20 0.44
HIF1A Q16665 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
ABCC3 O15438 1/20 0.43
ABCC4 O15439 1/20 0.43
CACNA1F O60840 1/20 0.43
ABCB11 O95342 1/20 0.43
ABCB1 P08183 1/20 0.43
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
TACR2 P21452 1/20 0.43
TBXAS1 P24557 1/20 0.43
OPRM1 P35372 1/20 0.43
DRD3 P35462 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13840781 0.79 CYP3A4 (0.54) CTSDCYP3A4LMNAUSP2CYP2D6
SCHEMBL2575749 0.79 CYP3A4 (0.54) CTSDCYP3A4LMNAUSP2CYP2D6
SCHEMBL4451153 0.78 CTSD (0.51) CTSDCYP3A4LMNAUSP2CYP2D6
SCHEMBL2577715 0.74 CYP3A4 (0.41) CTSDCYP3A4LMNAUSP2CYP2D6
SCHEMBL13825589 0.74 CYP3A4 (0.57) CTSDCYP3A4LMNAUSP2CYP2D6
SCHEMBL2576894 0.74 CYP3A4 (0.57) CTSDCYP3A4LMNAUSP2CYP2D6
SCHEMBL5689588 0.72 CYP3A4 (0.60) CTSDCYP3A4LMNAUSP2CYP2D6
SCHEMBL6224163 0.72 CYP3A4 (0.60) CTSDCYP3A4LMNAUSP2CYP2D6
SCHEMBL3041808 0.72 CYP3A4 (0.50) CTSDCYP3A4LMNAUSP2CYP2D6
SCHEMBL13219375 0.71 CYP3A4 (0.55) CTSDCYP3A4LMNAUSP2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5786483-A α-and β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors G. D. SEARLE & CO. (US) 1998-07-28 US claimed