SCHEMBL8624828

SCHEMBL8624828

CCCCN1CNS(=O)(=O)c2cnccc21

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 9/20 0.45
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 2/20 0.33
CA14 Q9ULX7 1/20 0.33
GAA P10253 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
TLR8 Q9NR97 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP19A1 P11511 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8623980 0.92 GRIA2 (0.47) GRIA2CA12CA1CA2CA9
SCHEMBL8625419 0.87 GRIA2 (0.58) GRIA2CA12CA1CA2CA9
SCHEMBL8561528 0.80 GRIA2 (0.50) GRIA2CA12CA1CA2CA9
SCHEMBL8625722 0.78 GRIA2 (0.42) GRIA2CA12CA1CA2CA9
SCHEMBL8556566 0.73 GRIA2 (0.35) GRIA2CA12CA1CA2CA9
SCHEMBL14415245 0.73 GRIA2 (0.51) GRIA2CA12CA1CA2CA9
SCHEMBL8627050 0.72 GRIA2 (0.38) GRIA2CA12CA1CA2CA9
SCHEMBL18186896 0.71 PIK3CD (0.39) GRIA2CA12CA1CA2CA9
SCHEMBL28750433 0.69 GRIA2 (0.42) GRIA2MEN1KMT2A
SCHEMBL8624379 0.68 CA12 (0.32) GRIA2CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618209-B1 Pyridothiadiazines, processes for their preparation and pharmaceutical compositions containing them ADIR (FR) 1998-12-23 EP disclosed
US-5459138-A Dysfunctions of glutamatergic neurotransmission associated with learning and memory ADIR ET COMPAGNIE (FR) 1995-10-17 US disclosed
EP-0618209-A1 Pyridothiadiazines, processes for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1994-10-05 EP disclosed