SCHEMBL8627744

SCHEMBL8627744

COc1ccc(N2CCN(CCN(C)C(=O)c3ccc4c(c3)CCOC4)CC2)cc1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 4/20 0.51
POLB P06746 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
DRD2 P14416 6/20 0.39
HTR1D P28221 5/20 0.39
HTR2A P28223 5/20 0.39
HTR1A P08908 3/20 0.39
SUV39H2 Q9H5I1 2/20 0.39
MAPT P10636 2/20 0.39
TSHR P16473 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CCR3 P51677 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTR1B P28222 1/20 0.38
DRD3 P35462 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549609 0.87 DRD4 (0.58) DRD4POLBMEN1KMT2ADRD2
SCHEMBL8550252 0.87 DRD4 (0.59) DRD4POLBDRD2HTR2AHTR1A
SCHEMBL8551575 0.84 DRD4 (0.48) DRD4DRD2HTR1DHTR2AHTR1A
SCHEMBL8550687 0.84 DRD4 (0.48) DRD4POLBKMT2ADRD2HTR1D
SCHEMBL8549471 0.84 DRD4 (0.48) DRD4DRD2HTR1DHTR2AHTR1A
SCHEMBL8553551 0.84 DRD4 (0.48) DRD4DRD2HTR1DHTR2AHTR1A
SCHEMBL8549399 0.84 CCR3 (0.56) DRD4KMT2ADRD2HTR1AMAPT
SCHEMBL8550036 0.83 DRD4 (0.47) DRD4POLBMEN1KMT2ADRD2
SCHEMBL8549100 0.83 DRD4 (0.47) DRD4MEN1KMT2ADRD2HTR1D
SCHEMBL8549415 0.82 DRD4 (0.49) DRD4MEN1KMT2ADRD2HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed