SCHEMBL8628513

SCHEMBL8628513

COC1CCC(CC(=O)N(C)C)c2cc(Cl)ccc2N1C(=O)c1ccc(NC(=O)c2ccccc2Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 5/20 0.44
AVPR2 P30518 4/20 0.44
HSD11B1 P28845 3/20 0.41
CHRM1 P11229 2/20 0.39
ABCB11 O95342 1/20 0.39
ADRB2 P07550 1/20 0.39
HTR1A P08908 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
TBXA2R P21731 1/20 0.39
HTR2C P28335 1/20 0.39
HRH1 P35367 1/20 0.39
OPRM1 P35372 1/20 0.39
GLP1R P43220 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39
GPR119 Q8TDV5 1/20 0.39
SPTLC2 O15270 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM3 P20309 1/20 0.39
TAS1R3 Q7RTX0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8627201 0.91 AVPR1A (0.46) AVPR1AAVPR2HSD11B1CHRM1ABCB11
SCHEMBL8632671 0.90 AVPR2 (0.44) AVPR1AAVPR2HSD11B1CHRM1ABCB11
Hydrochloric Acid SCHEMBL8634418 0.89 AVPR2 (0.41) AVPR1AAVPR2HSD11B1CHRM1ABCB11
SCHEMBL8635106 0.89 AVPR2 (0.43) AVPR1AAVPR2HSD11B1CHRM1ABCB11
SCHEMBL8630871 0.87 AVPR2 (0.44) AVPR1AAVPR2HSD11B1CHRM1ABCB11
Hydrochloric Acid SCHEMBL8634086 0.86 AVPR2 (0.43) AVPR1AAVPR2HSD11B1CHRM1ABCB11
SCHEMBL8629370 0.85 CHRM1 (0.48) AVPR1AAVPR2HSD11B1CHRM1ABCB11
SCHEMBL8630730 0.84 AVPR2 (0.47) AVPR1AAVPR2CHRM1ABCB11ADRB2
SCHEMBL8627097 0.84 SPTLC2 (0.51) AVPR1AAVPR2HSD11B1CHRM1ABCB11
SCHEMBL8632047 0.84 AVPR2 (0.43) AVPR1AAVPR2HSD11B1CHRM1ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US claimed