SCHEMBL8628631

SCHEMBL8628631

Nc1nc(CCC(N)C(=O)O)nc2[nH]cnc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 2/20 0.35
CYP3A4 P08684 1/20 0.35
SLC7A5 Q01650 1/20 0.35
ARG1 P05089 1/20 0.34
GRIK1 P39086 1/20 0.33
GRIA1 P42261 1/20 0.33
GRIA2 P42262 1/20 0.33
GRIA3 P42263 1/20 0.33
GRIA4 P48058 1/20 0.33
GRIK2 Q13002 1/20 0.33
GRIK3 Q13003 1/20 0.33
GRM8 O00222 1/20 0.33
GRM4 Q14833 1/20 0.33
GRM6 O15303 2/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
ALOX15 P16050 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11222090 0.80 PDPK1 (0.32)
SCHEMBL19839 0.79 CDK1 (0.36) ADORA2AADORA1
SCHEMBL8628643 0.79 PDPK1 (0.45) GRM2CYP1A2
SCHEMBL8592141 0.77 CYP1A2 (0.44) CYP3A4CYP1A2CYP2C19
SCHEMBL10357383 0.77 ADORA2A (0.34) ADORA2AADORA1
SCHEMBL5322828 0.77 CYP3A4 (0.38) GRM2CYP3A4SLC7A5ARG1GRIK1
SCHEMBL10361595 0.76 TBXAS1 (0.43)
SCHEMBL6379581 0.75 HRH2 (0.37)
SCHEMBL2060117 0.75 KDM4E (0.35) KMT2AADORA2AADORA1
SCHEMBL17165345 0.75 HTT (0.41) CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5705333-A Peptide-based nucleic acid mimics(PENAMS) THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1998-01-06 US disclosed