SCHEMBL8628960

SCHEMBL8628960

O=c1[nH]nc(C(C(OC(CO)(CO)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)c2ccccc2)N2CCCCC2)[nH]1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 18/20 0.43
TACR2 P21452 1/20 0.35
TACR3 P29371 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8628957 0.73 TACR1 (0.44) TACR1TACR2TACR3
SCHEMBL6938384 0.72 TACR1 (0.62) TACR1
SCHEMBL6486909 0.60 TACR1 (1.00) TACR1
SCHEMBL548109 0.57 SLC6A9 (0.49) TACR1
SCHEMBL16226493 0.56 KCNA5 (1.00)
SCHEMBL16227209 0.56 KCNA5 (1.00)
SCHEMBL16227210 0.56 KCNA5 (1.00)
SCHEMBL11866514 0.55 KCNA5 (0.68)
SCHEMBL31010271 0.54 KCNA5 (0.77)
SCHEMBL14033674 0.54 IDO1 (0.54) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760018-A Gem-disubstituted azacyclic tachykinin antagonists MERCK SHARP & DOHME LTD. (GB) 1998-06-02 US disclosed