SCHEMBL8630644

SCHEMBL8630644

CCOC(=O)c1csc(Cl)c1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.48
GRM6 O15303 1/20 0.43
CYP4F2 P78329 1/20 0.43
CYP4A11 Q02928 1/20 0.43
BAZ2B Q9UIF8 1/20 0.43
BAZ2A Q9UIF9 1/20 0.43
ALDH1A1 P00352 3/20 0.42
HSD17B10 Q99714 1/20 0.42
MAPT P10636 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
MAPK1 P28482 2/20 0.41
GAA P10253 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
CASP1 P29466 1/20 0.41
PRKCZ Q05513 1/20 0.41
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11484618 0.81 TSHR (0.52) TSHRALDH1A1HSD17B10MAPTMEN1
SCHEMBL6030900 0.80 TSHR (0.50) TSHRALDH1A1HSD17B10MAPTMEN1
SCHEMBL21543956 0.79 MAPT (0.53) TSHRALDH1A1HSD17B10MAPTMEN1
SCHEMBL3207148 0.78 CA1 (0.49) TSHRALDH1A1HSD17B10MAPTMEN1
SCHEMBL3879287 0.77 TSHR (0.47) TSHRALDH1A1HSD17B10MAPTMEN1
SCHEMBL18430422 0.77 ALDH1A1 (0.47) TSHRALDH1A1HSD17B10MAPTMEN1
SCHEMBL29474952 0.76 ALDH1A1 (0.50) TSHRALDH1A1HSD17B10MAPTMEN1
SCHEMBL28618971 0.75 TSHR (0.53) TSHRGRM6CYP4F2CYP4A11BAZ2B
SCHEMBL8632005 0.75 DAO (0.42) TSHRALDH1A1MAPTMEN1KMT2A
SCHEMBL18499644 0.75 GSK3B (0.40) ALDH1A1MAPTMEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5840917-A ADMINISTERING TO MAMMAL TO ERADICATE HELICOBACTER PYLORI TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-11-24 US disclosed
WO-1998042347-A1 PHARMACEUTICAL COMPOSITION CONTAINING A PHOSPHORYLAMIDE AND AN AYNTIBIOTIC TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-10-01 WO disclosed
EP-0852498-A1 PHOSPHORYLAMIDES, THEIR PREPARATION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-07-15 EP disclosed
WO-1997011705-A1 PHOSPHORYLAMIDES, THEIR PREPARATION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-04-03 WO disclosed