SCHEMBL8630765

SCHEMBL8630765

COc1cc(NC(=O)c2ccccc2Cl)ccc1C(=O)N1c2ccc(Cl)cc2CCCC1OCCSc1ncc[nH]1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 6/20 0.40
TP53 P04637 2/20 0.37
LMNA P02545 1/20 0.37
AVPR2 P30518 3/20 0.37
HSD17B10 Q99714 1/20 0.37
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MEN1 O00255 1/20 0.36
AVPR1A P37288 2/20 0.36
PTGS2 P35354 1/20 0.36
MAPT P10636 1/20 0.35
EGFR P00533 1/20 0.35
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8628611 0.91 GRM4 (0.42) GRM4TP53LMNAAVPR2HSD17B10
SCHEMBL8628510 0.87 GRM4 (0.40) GRM4TP53LMNAAVPR2HSD17B10
SCHEMBL8631655 0.87 GRM4 (0.40) GRM4TP53LMNAAVPR2KMT2A
SCHEMBL8634439 0.87 GRM4 (0.39) GRM4TP53LMNAAVPR2HSD17B10
SCHEMBL4684140 0.84 AVPR2 (0.46) GRM4AVPR2AVPR1A
SCHEMBL8627405 0.84 GRM4 (0.41) GRM4TP53LMNAAVPR2HSD17B10
SCHEMBL8630997 0.83 GRM4 (0.42) GRM4TP53LMNAAVPR2KMT2A
SCHEMBL8628504 0.83 GRM4 (0.42) GRM4TP53LMNAAVPR2HSD17B10
Hydrochloric Acid SCHEMBL8630791 0.81 GRM4 (0.41) GRM4TP53LMNAAVPR2HSD17B10
SCHEMBL8628615 0.81 GRM4 (0.40) GRM4TP53LMNAAVPR2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed