SCHEMBL8631041

SCHEMBL8631041

C#Cc1ccc2c(c1)C(C)(C)CC(=O)N2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 2/20 0.48
RARG P13631 2/20 0.48
HDAC3 O15379 6/20 0.43
HDAC4 P56524 6/20 0.43
HDAC1 Q13547 6/20 0.43
HDAC2 Q92769 6/20 0.43
HDAC8 Q9BY41 6/20 0.43
HDAC6 Q9UBN7 6/20 0.43
HDAC9 Q9UKV0 6/20 0.43
RARA P10276 1/20 0.36
PGR P06401 6/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
AHR P35869 3/20 0.33
CMA1 P23946 2/20 0.33
CYP46A1 Q9Y6A2 1/20 0.32
EIF2AK2 P19525 1/20 0.32
BACE1 P56817 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8630760 0.88 RARB (0.61) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL8629043 0.80 RARB (0.50) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL2242664 0.77 CYP1A2 (0.49) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL8867050 0.76 RARB (0.81) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL23078930 0.76 HDAC3 (0.49) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL248152 0.76 CMA1 (0.54) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL12072390 0.76 HDAC3 (0.46) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL1771822 0.76 CA9 (0.49) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL5643759 0.76 PGR (0.51) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL17675519 0.76 HDAC3 (0.46) RARBRARGHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825986-A1 QUINOLYL-ETHYNYL DERIVATIVES HAVING RETINOID-LIKE ACTIVITY Allergan (US) 1998-03-04 EP disclosed
US-5616712-A SKIN DISORDERS; ANTICARCINOGENIC AND -INFLAMMATORY AGENTS; AUTOIMMUNE DISEASES; ALLERGAN (US) 1997-04-01 US disclosed
WO-1996036609-A1 QUINOLYL-ETHYNYL DERIVATIVES HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1996-11-21 WO disclosed