SCHEMBL8632046

SCHEMBL8632046

CCOC(=O)COCc1nn[c]o1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.36
CA9 Q16790 2/20 0.36
MAPK1 P28482 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
ALDH1A1 P00352 4/20 0.34
KDM4E B2RXH2 3/20 0.34
HPGD P15428 2/20 0.34
HSD17B10 Q99714 2/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
GAA P10253 2/20 0.33
MGAM O43451 1/20 0.33
SI P14410 1/20 0.33
MGAM2 Q2M2H8 1/20 0.33
TSHR P16473 2/20 0.33
TRPA1 O75762 1/20 0.32
NPSR1 Q6W5P4 2/20 0.31
HRH3 Q9Y5N1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8629452 0.73 CA12 (0.39) CA12CA9MAPK1CA1CA2
SCHEMBL11416513 0.73 SMN1; SMN2 (0.39) CA12CA9MAPK1CA1CA2
SCHEMBL8628288 0.70 CA12 (0.36) CA12CA9MAPK1CA1CA2
SCHEMBL8626200 0.69 HRH3 (0.35) CA12CA9MAPK1CA1CA2
SCHEMBL3824014 0.68 TSHR (0.37) CA12CA9MAPK1CA1CA2
SCHEMBL2682415 0.68 GAA (0.60) CA12CA9CA1CA2ALDH1A1
SCHEMBL11119805 0.67 HSD17B10 (0.39) ALDH1A1KDM4EHSD17B10TP53MAPT
SCHEMBL2441045 0.67 CYP1A2 (0.38) CA12CA9MAPK1CA1CA2
SCHEMBL3829707 0.67 MAPK1 (0.35) CA12CA9MAPK1CA1CA2
SCHEMBL123093 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35754-E FOR TREATING BACTERIAL INFECTIONS HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US disclosed
US-5710146-A ANTIBIOTICS FOR BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1998-01-20 US disclosed
US-5089490-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1992-02-18 US disclosed
US-4758556-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1988-07-19 US disclosed
US-4399131-A Cephem derivatives HOECHST AG (DE) 1983-08-16 US disclosed
US-4278793-A ANTIBIOTICS, BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1981-07-14 US disclosed