SCHEMBL8633922

SCHEMBL8633922

CS(=O)(=O)C1=C(c2ccccc2)COC1=O

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.62
PTGS1 P23219 9/20 0.62
ALDH1A1 P00352 2/20 0.62
ABCB11 O95342 1/20 0.62
MT-CO2 P00403 1/20 0.62
HTR1A P08908 1/20 0.62
ADORA3 P0DMS8 1/20 0.62
MC4R P32245 1/20 0.62
KMT2A Q03164 2/20 0.56
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
POLB P06746 1/20 0.46
MAPT P10636 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Rofecoxib SCHEMBL4434618 0.77 PTGS2 (1.00) PTGS2PTGS1ALDH1A1ABCB11MT-CO2
SCHEMBL5858026 0.77 PTGS2 (1.00) PTGS2PTGS1ALDH1A1ABCB11MT-CO2
Rofecoxib SCHEMBL3050 0.77 PTGS2 (1.00) PTGS2PTGS1ALDH1A1ABCB11MT-CO2
Rofecoxib SCHEMBL14163950 0.77 PTGS2 (1.00) PTGS2PTGS1ALDH1A1ABCB11MT-CO2
Rofecoxib SCHEMBL28953295 0.76 PTGS2 (0.97) PTGS2PTGS1ALDH1A1ABCB11MT-CO2
Rofecoxib SCHEMBL7860859 0.76 PTGS2 (0.97) PTGS2PTGS1ALDH1A1ABCB11MT-CO2
Rofecoxib SCHEMBL6598209 0.76 PTGS2 (0.97) PTGS2PTGS1ALDH1A1ABCB11MT-CO2
SCHEMBL4390990 0.74 PTGS2 (0.58) PTGS2PTGS1ALDH1A1ABCB11MT-CO2
SCHEMBL7577906 0.73 PTGS2 (0.61) PTGS2PTGS1ALDH1A1ABCB11MT-CO2
SCHEMBL5071823 0.72 KMT2A (1.00) PTGS2PTGS1ALDH1A1ABCB11MT-CO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863891-A1 (METHYLSULFONYL)PHENYL-2-(5H)-FURANONES AS COX-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1998-09-16 EP claimed
WO-1997014691-A1 (METHYLSULFONYL)PHENYL-2-(5H)-FURANONES AS COX-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1997-04-24 WO claimed