SCHEMBL8634529

SCHEMBL8634529

N#Cc1c(N2CC3CCCNC3C2)c(F)cc2c(=O)c(OC(=O)OC3CC3)c[nH]c12

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
KMT2A Q03164 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7699514 1.00 KDM4E (0.44) KDM4EMEN1ALDH1A1HPGDKMT2A
SCHEMBL8319831 0.88 ALDH1A1 (0.47) KDM4EMEN1ALDH1A1HPGDKMT2A
SCHEMBL8363333 0.86 SSTR2 (0.35) KDM4EMEN1ALDH1A1HPGDKMT2A
SCHEMBL5166402 0.77
SCHEMBL7537093 0.74 KDM4E (0.61) KDM4EMEN1ALDH1A1HPGDKMT2A
SCHEMBL7541573 0.74 KDM4E (0.61) KDM4EMEN1ALDH1A1HPGDKMT2A
Hydrochloric Acid SCHEMBL7546889 0.73 KDM4E (0.62) KDM4EMEN1ALDH1A1HPGDKMT2A
SCHEMBL8366928 0.72 SSTR2 (0.33) KDM4EMEN1ALDH1A1HPGDKMT2A
SCHEMBL7248163 0.71 KDM4E (0.52) KDM4EMEN1ALDH1A1HPGDKMT2A
Trifluoroacetic Acid SCHEMBL7536833 0.71 KDM4E (0.57) KDM4EMEN1ALDH1A1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882049-A1 POSSIBLY SUBSTITUTED 8-CYANO-1-CYCLOPROPYL-7-(2,8-DIAZABICYCLO- 4.3.0]-NONAN-8-YL)-6-FLUORO-1,4-DIHYDRO-4-OXO-3-QUINOLIN CARBOXYLIC ACIDS AND THEIR DERIVATIVES BAYER AG (DE) 1998-12-09 EP claimed
WO-1997031001-A1 POSSIBLY SUBSTITUTED 8-CYANO-1-CYCLOPROPYL-7-(2,8-DIAZABICYCLO-[4.3.0]-NONAN-8-YL)-6-FLUORO-1,4-DIHYDRO-4-OXO-3-QUINOLIN CARBOXYLIC ACIDS AND THEIR DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 1997-08-28 WO claimed