SCHEMBL8634974

SCHEMBL8634974

CN(O)C(=S)SCC=Cn1cc(-c2ccc(Cl)cc2)c(-c2ccc(S(N)(=O)=O)cc2)n1.CN(O)C(=S)SCC=Cn1cc(-c2ccccc2)c(-c2ccc(S(N)(=O)=O)cc2)n1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 12/20 0.39
CA1 P00915 11/20 0.39
CA2 P00918 11/20 0.39
CA12 O43570 11/20 0.39
PTGS2 P35354 6/20 0.39
PTGS1 P23219 2/20 0.39
MAPK9 P45984 1/20 0.35
ENPP3 O14638 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6314715 0.97 CA1 (0.39) CA9CA1CA2CA12PTGS2
SCHEMBL6308406 0.96 CA9 (0.40) CA9CA1CA2CA12PTGS2
SCHEMBL8634963 0.92 PTGS2 (0.39) PTGS2PTGS1
SCHEMBL6309227 0.89 PTGS2 (0.39) PTGS2PTGS1
SCHEMBL6307645 0.88 PTGS2 (0.41) PTGS2PTGS1
SCHEMBL6744826 0.78 CA1 (0.46) CA9CA1CA2CA12PTGS2
SCHEMBL6747452 0.76 CA9 (0.43) CA9CA1CA2CA12PTGS2
SCHEMBL6746809 0.76 CA1 (0.39) CA9CA1CA2CA12PTGS2
SCHEMBL6314672 0.75 CA9 (0.40) CA9CA1CA2CA12PTGS2
SCHEMBL7777960 0.75 PTGS2 (0.49) CA9CA1CA2CA12PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828718-A1 HETEROCYCLO SUBSTITUTED HYDROXAMIC ACID DERIVATIVES AS CYCLOOXYGENASE-2 AND 5-LIPOXYGENASE INHIBITORS G.D. SEARLE & CO. (US) 1998-03-18 EP disclosed
WO-1996038418-A1 HETEROCYCLO SUBSTITUTED HYDROXAMIC ACID DERIVATIVES AS CYCLOOXYGENASE-2 AND 5-LIPOXYGENASE INHIBITORS G.D. SEARLE & CO. (US) 1996-12-05 WO disclosed