SCHEMBL8635868

SCHEMBL8635868

CN(O)C(=O)CCc1c(C(F)(F)F)nn(-c2ccc(S(N)(=O)=O)cc2)c1-c1ccc(F)cc1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.58
PTGS1 P23219 10/20 0.58
CA1 P00915 6/20 0.47
CA2 P00918 6/20 0.47
CA4 P22748 6/20 0.47
CA9 Q16790 6/20 0.47
CHRNA7 P36544 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8641301 0.91 PTGS2 (0.62) PTGS2PTGS1CA1CA2CA4
SCHEMBL8641056 0.89 PTGS2 (0.61) PTGS2PTGS1CA1CA2CA4
SCHEMBL8638794 0.88 PTGS2 (0.60) PTGS2PTGS1CA1CA2CA4
SCHEMBL8639285 0.86 PTGS2 (0.59) PTGS2PTGS1CA1CA2CA4
SCHEMBL5698589 0.85 PTGS2 (0.69) PTGS2PTGS1CA1CA2CA4
SCHEMBL8989633 0.80 PTGS2 (0.64) PTGS2PTGS1CA1CA2CA4
SCHEMBL8981470 0.80 PTGS2 (0.60) PTGS2PTGS1CA1CA2CA4
SCHEMBL6309336 0.77 CHRNA7 (0.60) PTGS2PTGS1CA1CA2CA9
SCHEMBL8989413 0.77 PTGS2 (0.57) PTGS2PTGS1CA1CA2CA4
SCHEMBL6013911 0.77 PTGS2 (0.81) PTGS2PTGS1CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5521207-A Substituted pyrazolyl benzenesulfonamide for the treatment of inflammation G.D. SEARLE & CO. (US) 1996-05-28 US disclosed
US-5516907-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-05-14 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5508426-A ANTIARTHRITIC AGENT G. D. SEARLE & CO. (US) 1996-04-16 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed
US-5466823-A Antiinflammatory agents; FDA Orange book listed patent for Celebrex G.D. SEARLE & CO. (US) 1995-11-14 US disclosed