SCHEMBL8635951

SCHEMBL8635951

O=S(=O)(Nn1nc(C(F)(F)F)cc1-c1cccnc1)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.54
PIK3CA P42336 1/20 0.43
PTGS1 P23219 3/20 0.42
HTR6 P50406 3/20 0.41
PDPK1 O15530 1/20 0.41
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.40
CKS1B P61024 1/20 0.38
SKP2 Q13309 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6520780 0.94 PTGS2 (0.48) PTGS2PIK3CAPTGS1HTR6PDPK1
SCHEMBL8640765 0.89 PTGS1 (0.51) PTGS2PTGS1PDPK1
SCHEMBL8638826 0.87 PTGS2 (0.49) PTGS2PIK3CAPTGS1PDPK1CYP2C9
SCHEMBL6515865 0.85 PDPK1 (0.45) PTGS2PIK3CAPTGS1PDPK1CYP3A4
SCHEMBL6517839 0.85 PTGS2 (0.47) PTGS2PIK3CAPTGS1HTR6PDPK1
SCHEMBL8641438 0.84 PTGS2 (0.43) PTGS2PTGS1PDPK1TSHRCYP3A4
SCHEMBL8641774 0.83 PTGS2 (0.41) PTGS2PTGS1PDPK1TSHRKMT2A
SCHEMBL8637254 0.82 PTGS2 (0.53) PTGS2PTGS1PDPK1
SCHEMBL8643941 0.82 PTGS2 (0.42) PTGS2PTGS1PDPK1
SCHEMBL8641577 0.82 PTGS2 (0.49) PTGS2PTGS1PDPK1KMT2ACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed