SCHEMBL8636808

SCHEMBL8636808

CCc1c(C(=O)O)nn(-c2ccc(S(N)(=O)=O)cc2)c1-c1ccc(Cl)cc1

nearest known ligand 0.74

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.74
PTGS1 P23219 8/20 0.67
CA1 P00915 6/20 0.64
CA2 P00918 6/20 0.64
CA4 P22748 6/20 0.64
CA9 Q16790 6/20 0.64
CHRNA7 P36544 4/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6341812 0.92 PTGS2 (0.71) PTGS2PTGS1CA1CA2CA4
SCHEMBL28248642 0.90 PTGS2 (0.58) PTGS2PTGS1CA1CA2CA4
SCHEMBL6349532 0.90 PTGS2 (0.69) PTGS2PTGS1CA1CA2CA4
SCHEMBL6351372 0.89 PTGS2 (0.67) PTGS2PTGS1CA1CA2CA4
SCHEMBL6353455 0.89 PTGS2 (0.70) PTGS2PTGS1CA1CA2CA4
SCHEMBL6341478 0.85 PTGS2 (0.79) PTGS2PTGS1CA1CA2CA4
SCHEMBL6339325 0.85 PTGS2 (1.00) PTGS2PTGS1CA1CA2CA4
SCHEMBL8120953 0.84 PTGS2 (0.72) PTGS2PTGS1CA1CA2CA4
SCHEMBL3867425 0.83 PTGS2 (0.63) PTGS2PTGS1CA1CA2CA4
SCHEMBL6350079 0.83 PTGS2 (0.79) PTGS2PTGS1CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5563165-A PROSTAGLANDIN INHIBITOR; FDA ORANGE BOOK LISTED PATENT FOR CELEBREX G. D. SEARL & CO. (US) 1996-10-08 US disclosed
US-5521207-A Substituted pyrazolyl benzenesulfonamide for the treatment of inflammation G.D. SEARLE & CO. (US) 1996-05-28 US disclosed
US-5516907-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-05-14 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5508426-A ANTIARTHRITIC AGENT G. D. SEARLE & CO. (US) 1996-04-16 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed
US-5466823-A Antiinflammatory agents; FDA Orange book listed patent for Celebrex G.D. SEARLE & CO. (US) 1995-11-14 US disclosed