SCHEMBL8637843

SCHEMBL8637843

O=C(CCCN1CCN(c2ccncc2)CC1)Oc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 12/20 0.60
HRH1 P35367 6/20 0.60
HRH2 P25021 2/20 0.60
HTR1A P08908 2/20 0.51
DRD2 P14416 1/20 0.51
HTR2A P28223 1/20 0.51
DRD3 P35462 1/20 0.51
TMEM97 Q5BJF2 1/20 0.51
SIGMAR1 Q99720 1/20 0.51
ALDH1A1 P00352 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
TSHR P16473 1/20 0.51
MAPK1 P28482 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
HIF1A Q16665 1/20 0.51
DRD4 P21917 1/20 0.51
SLC6A4 P31645 1/20 0.51
HTR7 P34969 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8630602 0.96 HRH3 (0.59) HRH3HRH1HRH2HTR1AALDH1A1
SCHEMBL8634144 0.88 HRH3 (0.57) HRH3HRH1HRH2
SCHEMBL8701067 0.85 HRH3 (0.58) HRH3HRH1HRH2DRD4SLC6A4
SCHEMBL8634523 0.83 KCNH2 (0.52) HRH3HRH1HRH2ALDH1A1CYP2D6
SCHEMBL8635007 0.82 DRD4 (0.60) HRH3HRH1HRH2DRD4SLC6A4
SCHEMBL8632823 0.81 FAAH (0.44) HRH3HRH1HRH2HTR1ADRD2
Hydrochloric Acid SCHEMBL27454125 0.80 DRD4 (0.58) HRH3HRH1HRH2DRD4SLC6A4
Hydrochloric Acid SCHEMBL8838070 0.79 HRH3 (0.56) HRH3HRH1HRH2HTR2ADRD4
SCHEMBL8630675 0.78 CYP2C9 (0.40) HRH3HRH1HRH2ALDH1A1CYP2D6
SCHEMBL8681193 0.78 CYP2C9 (0.40) HRH3HRH1HRH2ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US claimed
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed
CN-1120334-A Heterocyclic derivatives as platelet aggregation inhibitors ZENECA LTD (GB) 1996-04-10 CN disclosed