SCHEMBL8638779

SCHEMBL8638779

COC(=O)Cc1ccc(-n2nc(C(F)(F)F)cc2-c2ccc(S(C)(=O)=O)cc2)cc1

nearest known ligand 0.79

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.79
PTGS1 P23219 3/20 0.66
CYP2C9 P11712 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8645174 0.89 PTGS2 (1.00) PTGS2PTGS1CYP2C9
SCHEMBL9089381 0.85 PTGS2 (0.79) PTGS2PTGS1CYP2C9
SCHEMBL16426376 0.84 PTGS2 (0.76) PTGS2PTGS1CYP2C9
SCHEMBL8953880 0.84 PTGS2 (0.81) PTGS2PTGS1CYP2C9
SCHEMBL27531784 0.83 PTGS2 (0.75) PTGS2PTGS1CYP2C9
SCHEMBL7461840 0.82 PTGS2 (0.81) PTGS2PTGS1CYP2C9
SCHEMBL7466325 0.81 PTGS2 (0.80) PTGS2PTGS1CYP2C9
SCHEMBL8925698 0.81 PTGS2 (0.71) PTGS2PTGS1CYP2C9
SCHEMBL7457684 0.81 PTGS2 (0.74) PTGS2PTGS1CYP2C9
SCHEMBL8925277 0.81 PTGS2 (0.79) PTGS2PTGS1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0856000-A1 1,3,5-TRISUBSTITUTED PYRAZOLES FOR TREAMENT OF INFLAMMATION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-08-05 EP disclosed
WO-1997013755-A1 1,3,5-TRISUBSTITUTED PYRAZOLES FOR TREAMENT OF INFLAMMATION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-04-17 WO disclosed