SCHEMBL8639159

SCHEMBL8639159

COc1cc(Cl)ccc1-c1cc(C(F)(F)F)nn1-c1ccccc1S(N)(=O)=O

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.57
PTGS1 P23219 7/20 0.52
PDPK1 O15530 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8639427 0.89 PTGS2 (0.61) PTGS2PTGS1
SCHEMBL8690936 0.89 PTGS2 (0.58) PTGS2PTGS1
SCHEMBL8636819 0.89 PTGS2 (0.72) PTGS2PTGS1
SCHEMBL8640004 0.87 PTGS2 (0.55) PTGS2PTGS1PDPK1
SCHEMBL8635927 0.87 PTGS2 (0.68) PTGS2PTGS1PDPK1
SCHEMBL8637080 0.85 PTGS2 (0.57) PTGS2PTGS1PDPK1
SCHEMBL8641744 0.84 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL6340153 0.83 PTGS2 (0.76) PTGS2PTGS1PDPK1
SCHEMBL8689327 0.82 PTGS2 (0.57) PTGS2PTGS1PDPK1
SCHEMBL8689333 0.82 PTGS2 (0.62) PTGS2PTGS1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed