SCHEMBL8639175

SCHEMBL8639175

Cc1cc(-c2ccccc2)n(-c2ccccc2S(N)(=O)=O)n1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.64
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
ALOX5 P09917 1/20 0.54
ALDH1A1 P00352 4/20 0.50
HPGD P15428 2/20 0.50
CA1 P00915 3/20 0.48
CA2 P00918 3/20 0.48
CA9 Q16790 3/20 0.48
CA12 O43570 2/20 0.48
CYP2C9 P11712 2/20 0.45
F10 P00742 3/20 0.45
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C19 P33261 1/20 0.43
RECQL P46063 1/20 0.43
PTGS1 P23219 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8422373 0.84 CYP2C9 (0.55) PTGS2ALDH1A1CA1CA2CA9
SCHEMBL8689524 0.84 PTGS2 (0.45) PTGS2ALOX5ALDH1A1CA1CA2
SCHEMBL8691378 0.83 PTGS2 (0.44) PTGS2NPC1RAB9AALOX5ALDH1A1
SCHEMBL8689301 0.83 PTGS2 (0.44) PTGS2ALDH1A1CA1CA2CA9
SCHEMBL8691619 0.83 PTGS2 (0.44) PTGS2ALDH1A1CA1CA2CA9
SCHEMBL8688892 0.81 PTGS2 (0.51) PTGS2ALOX5ALDH1A1CA1CA2
SCHEMBL8691565 0.81 PTGS2 (0.42) PTGS2ALOX5ALDH1A1CA1CA2
SCHEMBL6406740 0.80 CA9 (0.66) PTGS2CA1CA2CA9
SCHEMBL8688836 0.80 PTGS2 (0.66) PTGS2ALOX5ALDH1A1CA1CA2
SCHEMBL8420750 0.80 CYP2C9 (0.63) PTGS2NPC1RAB9AALOX5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed