SCHEMBL8639593

SCHEMBL8639593

CCCCS(=O)(=O)Nn1c(C(=O)O)cc2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.47
DAO P14920 1/20 0.44
CCR2 P41597 3/20 0.43
ALDH1A1 P00352 3/20 0.43
TSHR P16473 1/20 0.43
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41
PLA2G4A P47712 1/20 0.41
CNR2 P34972 3/20 0.39
OXER1 Q8TDS5 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5728166 0.78 MCL1 (0.50) MCL1DAOCCR2ALDH1A1TSHR
SCHEMBL5008889 0.78 MCL1 (0.50) MCL1DAOCCR2ALDH1A1TSHR
SCHEMBL7208143 0.76 DAO (0.51) MCL1DAOCCR2ALDH1A1TSHR
SCHEMBL10757133 0.72 ALDH1A1 (0.66) MCL1DAOCCR2ALDH1A1TSHR
SCHEMBL6682164 0.70 ALDH1A1 (0.64) MCL1DAOCCR2ALDH1A1CYP1A2
SCHEMBL10379817 0.70 DAO (0.59) MCL1DAOCCR2ALDH1A1TSHR
SCHEMBL8551062 0.70 MCL1 (0.57) MCL1DAOCCR2ALDH1A1TSHR
SCHEMBL6685154 0.70 MCL1 (0.57) MCL1DAOCCR2ALDH1A1TSHR
SCHEMBL10762525 0.69 ALDH1A1 (0.63) MCL1DAOCCR2ALDH1A1CYP1A2
SCHEMBL8242370 0.69 ALDH1A1 (0.63) MCL1DAOCCR2ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed