SCHEMBL8640586

SCHEMBL8640586

NNC(=O)Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.55
BACE1 P56817 1/20 0.48
BACE2 Q9Y5Z0 1/20 0.48
ALDH1A1 P00352 1/20 0.47
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
KDM4E B2RXH2 1/20 0.46
PSEN1 P49768 2/20 0.46
PSEN2 P49810 2/20 0.46
APH1B Q8WW43 2/20 0.46
NCSTN Q92542 2/20 0.46
APH1A Q96BI3 2/20 0.46
PSENEN Q9NZ42 2/20 0.46
CYP2D6 P10635 1/20 0.46
IDO1 P14902 2/20 0.46
CES2 O00748 1/20 0.45
LMNA P02545 1/20 0.45
RXRA P19793 1/20 0.45
RXRB P28702 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867356 0.82 MEN1 (0.68) ALDH1A1MEN1MAPTKMT2AKDM4E
Hydrochloric Acid SCHEMBL6208799 0.81 TACR1 (0.52) TACR1BACE1BACE2MEN1MAPT
SCHEMBL19301048 0.81 TACR1 (0.56) TACR1BACE1BACE2MEN1MAPT
SCHEMBL714137 0.81 HDAC1 (0.63) BACE1BACE2ALDH1A1KDM4EHDAC1
SCHEMBL13753363 0.80 TACR1 (0.58) TACR1BACE1BACE2ALDH1A1MEN1
SCHEMBL12471510 0.80 TACR1 (0.58) TACR1BACE1BACE2MEN1MAPT
SCHEMBL2484345 0.80 IDO1 (0.48) TACR1IDO1CES2RXRARXRB
SCHEMBL6865708 0.79 CES2 (0.52) TACR1MAPTIDO1CES2LMNA
Hydrochloric Acid SCHEMBL3143821 0.78 IDO1 (0.50) TACR1IDO1CES2RXRARXRB
Hydrochloric Acid SCHEMBL3152131 0.78 IDO1 (0.50) TACR1IDO1CES2RXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5710161-A Triazole derivatives and their use as therapeutic agents MERCK, SHARP & DOHME, LTD. (GB) 1998-01-20 US disclosed