SCHEMBL8640609

SCHEMBL8640609

Cc1ccc(Cn2nc(Br)c([N+](=O)[O-])c2NCc2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.50
MAPT P10636 4/20 0.45
ALDH1A1 P00352 3/20 0.43
HTT P42858 3/20 0.43
NPC1 O15118 1/20 0.43
CYP3A4 P08684 1/20 0.43
HPGD P15428 1/20 0.42
MC4R P32245 1/20 0.40
NR1H4 Q96RI1 2/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KDM4E B2RXH2 1/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA13 Q8N1Q1 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8919318 0.93 HTT (0.44) SMN1; SMN2MAPTALDH1A1HTTCYP3A4
SCHEMBL8641624 0.90 MAPT (0.46) SMN1; SMN2MAPTALDH1A1HTTNPC1
SCHEMBL9088185 0.88 EGFR (0.50) SMN1; SMN2MAPTALDH1A1HTTNPC1
SCHEMBL6755732 0.87 MAPT (0.42) SMN1; SMN2MAPTALDH1A1HTTCYP3A4
SCHEMBL8920720 0.85 MAPT (0.41) SMN1; SMN2MAPTALDH1A1HTTCYP3A4
SCHEMBL8920097 0.85 CYP3A4 (0.44) SMN1; SMN2MAPTALDH1A1HTTCYP3A4
SCHEMBL1026866 0.84 KDM4E (0.45) SMN1; SMN2MAPTALDH1A1HTTCYP3A4
SCHEMBL6755855 0.83 HTT (0.47) SMN1; SMN2MAPTALDH1A1HTTCYP3A4
SCHEMBL8922319 0.82 MAPT (0.43) SMN1; SMN2MAPTALDH1A1HTTCYP3A4
SCHEMBL9087932 0.82 MAPT (0.48) SMN1; SMN2MAPTALDH1A1NR1H4L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5718731-A Oxidation hair dye composition based on 4,5-diaminopyrazole and m-phenylenediamine derivatives WELLA AKTIENGESELLSCHAFT (DE) 1998-02-17 US disclosed
EP-0692245-B1 Oxidation hair dye containing 4,5-diaminopyrazole derivatives and m-phenylendiamine derivatives WELLA AG (DE) 1997-05-02 EP disclosed
US-5534267-A Composition for the oxidative dyeing of hair containing 4,5-diaminopyrazole derivatives as well as new 4,5-diaminopyrazole derivatives and process for their synthesis WELLA AKTIENGESELLSCHAFT (DE) 1996-07-09 US disclosed
EP-0692245-A1 Oxidation hair dye containing 4,5-diaminopyrazole derivatives and m-phenylendiamine derivatives Wella Aktiengesellschaft (DE) 1996-01-17 EP disclosed
EP-0618903-A1 OXIDATION HAIR DYE CONTAINING 4,5-DIAMINOPYRAZOLE DERIVATIVES AND NOVEL 4,5-DIAMINOPYRAZOLE DERIVATIVES AND PROCESS FOR THEIR PRODUCTION Wella Aktiengesellschaft (DE) 1994-10-12 EP disclosed
WO-1994008970-A1 OXIDATION HAIR DYE CONTAINING 4,5-DIAMINOPYRAZOLE DERIVATIVES AND NOVEL 4,5-DIAMINOPYRAZOLE DERIVATIVES AND PROCESS FOR THEIR PRODUCTION WELLA AKTIENGESELLSCHAFT (DE) 1994-04-28 WO disclosed