SCHEMBL8640762

SCHEMBL8640762

NS(=O)(=O)c1ccccc1-n1nc(C(F)(F)F)cc1-c1ccc(O)c(O)c1

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 6/20 0.53
PTGS2 P35354 13/20 0.52
PTGS1 P23219 5/20 0.52
CYP2C9 P11712 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8662511 0.90 PTGS2 (0.50) PDPK1PTGS2PTGS1CYP2C9
SCHEMBL8688454 0.90 PTGS2 (0.52) PDPK1PTGS2PTGS1CYP2C9
SCHEMBL8638820 0.90 PDPK1 (0.57) PDPK1PTGS2PTGS1CYP2C9
SCHEMBL8637585 0.87 PDPK1 (0.69) PDPK1PTGS2PTGS1CYP2C9
SCHEMBL8640768 0.87 PTGS2 (0.67) PDPK1PTGS2PTGS1CYP2C9
SCHEMBL8638225 0.86 PDPK1 (0.71) PDPK1PTGS2PTGS1CYP2C9
SCHEMBL8641581 0.86 PTGS2 (0.65) PDPK1PTGS2PTGS1CYP2C9
SCHEMBL5694290 0.86 PTGS2 (0.65) PDPK1PTGS2PTGS1CYP2C9
SCHEMBL8643577 0.86 PTGS2 (0.65) PDPK1PTGS2PTGS1CYP2C9
SCHEMBL8641602 0.85 PTGS2 (0.53) PDPK1PTGS2PTGS1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed