SCHEMBL8640766

SCHEMBL8640766

C=C(C)C(=O)c1cccnc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.57
GAA P10253 3/20 0.57
APP P05067 1/20 0.57
HCAR3 P49019 1/20 0.57
HCAR2 Q8TDS4 1/20 0.57
F7 P08709 1/20 0.55
F3 P13726 1/20 0.55
SARM1 Q6SZW1 1/20 0.55
SIRT2 Q8IXJ6 1/20 0.55
SIRT6 Q8N6T7 1/20 0.55
SIRT1 Q96EB6 1/20 0.55
SIRT3 Q9NTG7 1/20 0.55
SIRT5 Q9NXA8 1/20 0.55
SIRT4 Q9Y6E7 1/20 0.55
HDAC1 Q13547 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
LMNA P02545 2/20 0.49
CYP1A2 P05177 2/20 0.49
CYP3A4 P08684 2/20 0.49
CYP11B1 P15538 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13271880 1.00 ALDH1A1 (0.57) ALDH1A1GAAAPPHCAR3HCAR2
SCHEMBL2690817 0.86 ALDH1A1 (0.63) ALDH1A1GAAAPPHCAR3HCAR2
SCHEMBL2784997 0.83 ALDH1A1 (0.71) ALDH1A1GAAAPPHCAR3HCAR2
SCHEMBL1642463 0.80 ALDH1A1 (0.52) ALDH1A1GAAAPPHCAR3HCAR2
SCHEMBL10860350 0.79 ALDH1A1 (0.65) ALDH1A1GAAAPPHCAR3HCAR2
SCHEMBL29496911 0.79
SCHEMBL1699 0.79
SCHEMBL1258378 0.79
SCHEMBL609057 0.79
SCHEMBL8039612 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857721-A1 ACRIDONE COMPOUNDS Eisai Co., Ltd. (JP) 1998-08-12 EP disclosed