SCHEMBL8640912

SCHEMBL8640912

OC[C@H]1O[C@@H](CI)C[C@@H]1OCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 3/20 0.54
SLC6A2 P23975 2/20 0.42
TSHR P16473 1/20 0.41
CYP2C19 P33261 1/20 0.41
TACR2 P21452 1/20 0.38
GYPA P02724 1/20 0.38
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
BCHE P06276 2/20 0.36
CTSV O60911 1/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
CTSC P53634 1/20 0.35
CTSF Q9UBX1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8647380 1.00 PDE4D (0.54) PDE4DSLC6A2TSHRCYP2C19TACR2
SCHEMBL10809088 0.81 PDE4D (0.61) PDE4DSLC6A2TSHRCYP2C19GYPA
SCHEMBL10803799 0.81 PDE4D (0.61) PDE4DSLC6A2TSHRCYP2C19GYPA
SCHEMBL8644844 0.80 PDE4D (0.56) PDE4DSLC6A2TSHRCYP2C19TACR2
SCHEMBL31556088 0.80 PDE4D (0.59) PDE4DSLC6A2GYPABCHEACHE
SCHEMBL10807993 0.78 PDE4D (0.54) PDE4DSLC6A2TSHRCYP2C19GYPA
SCHEMBL25084227 0.76 PDE4D (0.52) PDE4DSLC6A2TSHRCYP2C19GYPA
SCHEMBL9799958 0.76 PDE4D (0.55) PDE4DSLC6A2TSHRCYP2C19GYPA
SCHEMBL9432360 0.76 PDE4D (0.52) PDE4DSLC6A2TSHRCYP2C19GYPA
SCHEMBL11558436 0.75 PDE4D (0.45) PDE4DSLC6A2PSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750735-A CHEMICAL INTERMEDIATES FOR ANTIBIOTICS AMERICAN CYANAMID COMPANY (US) 1998-05-12 US disclosed
US-5744465-A Method of inhibiting a β-lactamase enzyme by administering novel 2-thiosubstituted carbapenems AMERICAN CYANAMID COMPANY (US) 1998-04-28 US disclosed
US-5623081-A USING BENZYLOXYACETALDEHYDE DIMETHYL ETHER, HALOGENATED 1-PHENYLMETHOXY-4-PENTEN-2-OL; CYCLIZATION LIN YANG-I (US) 1997-04-22 US disclosed
US-5602118-A A 2-((2-SUBSTITUTED ALKYL)FUR-3-YL)-THIO-),3-CARBOXY-2-CARBOPENEM DERIVATIVES; EFFECTIVE AGAINST BETA-LACTAM ANTIBIOTIC-RESISTANT BACTERIA AMERICAN CYANAMID COMPANY (US) 1997-02-11 US disclosed
EP-0617036-A2 Novel 2-thiosubstituted carbapenems AMERICAN CYANAMID COMPANY (US) 1994-09-28 EP disclosed