SCHEMBL8640966

SCHEMBL8640966

NS(=O)(=O)c1ccc(NC(=O)c2cc(-c3ccc(Cl)cc3)[nH]n2)cc1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.56
MEN1 O00255 3/20 0.56
CA2 P00918 8/20 0.56
CA1 P00915 7/20 0.56
CA9 Q16790 5/20 0.56
CA12 O43570 3/20 0.56
MAPK9 P45984 1/20 0.55
ALDH1A1 P00352 1/20 0.54
LMNA P02545 1/20 0.54
POLB P06746 1/20 0.54
CA4 P22748 2/20 0.54
CA7 P43166 1/20 0.54
CDK2 P24941 3/20 0.51
CDK1 P06493 2/20 0.51
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8691553 0.89 PTPN7 (0.54) KMT2AMEN1CA2CA1CA9
SCHEMBL8694108 0.89 CDK2 (0.64) KMT2AMEN1CA2CA1CA9
SCHEMBL8642022 0.89 CDK2 (0.64) KMT2AMEN1CA2CA1CA9
SCHEMBL8690975 0.89 KMT2A (0.57) KMT2AMEN1CA2CA1CA9
SCHEMBL8688552 0.86 CDK2 (0.52) KMT2ACA2CA1CA9CA12
SCHEMBL8688441 0.86 CDK2 (0.47) KMT2AMEN1CA2CA1CA9
SCHEMBL8691753 0.86 CDK2 (0.66) CA2CA1CA9CA12ALDH1A1
SCHEMBL20764122 0.84 NPC1 (0.52) MAPT
SCHEMBL8692528 0.83 CDK2 (0.54) KMT2AMEN1CA2CA1CA9
SCHEMBL8732480 0.82 KMT2A (0.47) KMT2AMEN1CA2CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed