SCHEMBL8688552

SCHEMBL8688552

COc1ccc(-c2cc(C(=O)Nc3ccc(S(N)(=O)=O)cc3)n[nH]2)cc1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 3/20 0.52
CDK1 P06493 2/20 0.52
CA1 P00915 12/20 0.51
CA2 P00918 12/20 0.51
CA9 Q16790 8/20 0.51
CA12 O43570 8/20 0.51
ALDH1A1 P00352 1/20 0.51
KMT2A Q03164 1/20 0.51
CA4 P22748 2/20 0.50
CA7 P43166 2/20 0.50
PTGS2 P35354 1/20 0.48
MAOB P27338 1/20 0.48
CA5A P35218 1/20 0.48
CA5B Q9Y2D0 1/20 0.48
CSNK2A2 P19784 1/20 0.47
CSNK2A1 P68400 1/20 0.47
TNIK Q9UKE5 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8691553 0.88 PTPN7 (0.54) CDK2CDK1CA1CA2CA9
SCHEMBL8640966 0.86 KMT2A (0.56) CDK2CDK1CA1CA2CA9
SCHEMBL8688685 0.85 CDK2 (0.54) CDK2CDK1CA1CA2CA9
SCHEMBL8692528 0.85 CDK2 (0.54) CDK2CDK1CA1CA2CA9
SCHEMBL8642022 0.85 CDK2 (0.64) CDK2CDK1CA1CA2CA9
SCHEMBL8694108 0.85 CDK2 (0.64) CDK2CDK1CA1CA2CA9
SCHEMBL8690975 0.85 KMT2A (0.57) CDK2CDK1CA1CA2CA9
SCHEMBL8732480 0.85 KMT2A (0.47) CDK2CDK1CA1CA2CA9
SCHEMBL8688441 0.85 CDK2 (0.47) CDK2CDK1CA1CA2CA9
SCHEMBL8691753 0.83 CDK2 (0.66) CDK2CDK1CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed