SCHEMBL8645113

SCHEMBL8645113

NC(=O)[C@H](NC=O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.44
CYP2D6 P10635 2/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
PDGFRA P16234 1/20 0.42
MAPK1 P28482 1/20 0.42
MAPKAPK2 P49137 1/20 0.42
RPS6KA1 Q15418 1/20 0.42
AURKB Q96GD4 1/20 0.42
CSNK1G1 Q9HCP0 1/20 0.42
EPHX1 P07099 2/20 0.42
KMT2A Q03164 2/20 0.41
CTSD P07339 1/20 0.41
BCAT2 O15382 1/20 0.41
TACR3 P29371 1/20 0.40
SRC P12931 1/20 0.39
LMNA P02545 1/20 0.39
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10402082 1.00 OPRK1 (0.44) OPRK1CYP2D6CYP3A4CYP2C9PDGFRA
SCHEMBL2777368 0.84 CYP2D6 (0.52) OPRK1CYP2D6MAPK1EPHX1KMT2A
SCHEMBL14871996 0.84 CYP2D6 (0.52) OPRK1CYP2D6MAPK1EPHX1KMT2A
SCHEMBL2478440 0.84 CYP2D6 (0.52) OPRK1CYP2D6MAPK1EPHX1KMT2A
SCHEMBL12174989 0.81 OPRK1 (0.47) OPRK1CYP2D6MAPK1EPHX1KMT2A
SCHEMBL10402081 0.81 OPRK1 (0.44) OPRK1CYP2D6MAPK1EPHX1KMT2A
SCHEMBL15359365 0.81 OPRK1 (0.47) OPRK1CYP2D6MAPK1EPHX1KMT2A
SCHEMBL12158471 0.78 OPRK1 (0.45) OPRK1CYP2D6CYP3A4EPHX1KMT2A
SCHEMBL11991382 0.78 KMT2A (0.61) OPRK1CYP2D6CYP3A4CYP2C9KMT2A
SCHEMBL8505416 0.78 KMT2A (0.61) OPRK1CYP2D6CYP3A4CYP2C9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5854268-A Azetidine, pyrrolidine and piperidine derivatives MERCK SHARP & DOHME, LTD. (GB) 1998-12-29 US disclosed