SCHEMBL8645966

SCHEMBL8645966

O=[N+]([O-])c1ccc2c(N3CCc4ccc(Cl)cc43)ncnc2c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.47
EGFR P00533 6/20 0.46
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
RPS6KB1 P23443 2/20 0.41
CSF1R P07333 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
PDGFRB P09619 1/20 0.41
DRD2 P14416 1/20 0.40
MAPT P10636 2/20 0.39
ACHE P22303 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
BACE1 P56817 1/20 0.39
AURKA O14965 1/20 0.39
LMNA P02545 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8649552 0.99 ROCK1 (0.46) ROCK1EGFRHTTSMN1; SMN2RPS6KB1
SCHEMBL8648167 0.92 ROCK1 (0.47) ROCK1EGFRHTTSMN1; SMN2RPS6KB1
SCHEMBL9115422 0.88 ROCK1 (0.44) ROCK1EGFRHTTSMN1; SMN2RPS6KB1
SCHEMBL9116362 0.88 EGFR (0.47) ROCK1EGFRHTTSMN1; SMN2CSF1R
SCHEMBL8650186 0.86 CYP1A2 (0.52) ROCK1EGFRHTTCSF1RCYP1A2
SCHEMBL8646578 0.83 EGFR (0.46) EGFRHTTCSF1RCYP1A2CYP2D6
Hydrochloric Acid SCHEMBL8647893 0.81 EGFR (0.47) ROCK1EGFRHTTSMN1; SMN2RPS6KB1
SCHEMBL8651028 0.81 EGFR (0.48) EGFRHTTSMN1; SMN2RPS6KB1CSF1R
SCHEMBL7499713 0.80 RPS6KB1 (0.44) ROCK1HTTSMN1; SMN2RPS6KB1CSF1R
SCHEMBL8650199 0.80 EGFR (0.49) ROCK1EGFRHTTCSF1RCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5736534-A HYPERPROLIFERATIVE DISEASES; INHIBITORS OF PROTEIN-TYROSINE KINASES SUCH AS EPIDERMAL GROWTH FACTOR RECEPTOR; BRAIN, LUNG, BREAST CANCER; PSORIASIS AND BENIGN PROSTATE HYPERPLASIA PFIZER INC. (US) 1998-04-07 US disclosed
CN-1141633-A 4-heterocyclic substituted quinazoline derivatives, process for their preparation and their use as anticancer agents PFIZER (US) 1997-01-29 CN disclosed