SCHEMBL8646304

SCHEMBL8646304

COc1cc2ncnc(N3CCc4cc(N)ccc43)c2cc1OC

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 6/20 0.75
CSF1R P07333 1/20 0.73
RET P07949 2/20 0.60
KDR P35968 2/20 0.60
KIF5B P33176 1/20 0.60
KIT P10721 3/20 0.56
ACHE P22303 6/20 0.54
BACE1 P56817 6/20 0.54
PDGFRB P09619 2/20 0.50
TUBB4A P04350 1/20 0.50
TUBB P07437 1/20 0.50
TUBA3C P0DPH7 1/20 0.50
TUBA1B P68363 1/20 0.50
TUBA4A P68366 1/20 0.50
TUBB4B P68371 1/20 0.50
TUBB3 Q13509 1/20 0.50
TUBB2A Q13885 1/20 0.50
TUBB8 Q3ZCM7 1/20 0.50
TUBA3E Q6PEY2 1/20 0.50
TUBA1A Q71U36 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8649920 0.99 EGFR (0.76) EGFRCSF1RRETKDRKIF5B
SCHEMBL8644637 0.91 EGFR (0.75) EGFRCSF1RRETKDRKIF5B
SCHEMBL8652258 0.88 EGFR (0.75) EGFRCSF1RRETKDRKIF5B
SCHEMBL9115430 0.88 EGFR (0.75) EGFRCSF1RRETKDRKIF5B
SCHEMBL8647385 0.87 EGFR (0.73) EGFRCSF1RRETKDRKIF5B
SCHEMBL8645023 0.87 EGFR (0.73) EGFRCSF1RRETKDRKIF5B
SCHEMBL6185124 0.86 EGFR (1.00) EGFRCSF1RRETKDRKIF5B
Hydrochloric Acid SCHEMBL6179838 0.85 EGFR (1.00) EGFRCSF1RRETKDRKIF5B
SCHEMBL9116168 0.83 EGFR (0.67) EGFRCSF1RRETKDRKIF5B
SCHEMBL8648530 0.83 EGFR (0.67) EGFRCSF1RRETKDRKIF5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5736534-A HYPERPROLIFERATIVE DISEASES; INHIBITORS OF PROTEIN-TYROSINE KINASES SUCH AS EPIDERMAL GROWTH FACTOR RECEPTOR; BRAIN, LUNG, BREAST CANCER; PSORIASIS AND BENIGN PROSTATE HYPERPLASIA PFIZER INC. (US) 1998-04-07 US disclosed
EP-0746554-A1 4-HETEROCYCLYL-SUBSTITUTED QUINAZOLINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS ANTI-CANCER AGENTS PFIZER INC. (US) 1996-12-11 EP disclosed
WO-1995023141-A1 4-HETEROCYCLYL-SUBSTITUTED QUINAZOLINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS ANTI-CANCER AGENTS PFIZER INC. (US) 1995-08-31 WO disclosed