SCHEMBL8647804

SCHEMBL8647804

CC(C)(C)[Si](C)(C)Oc1ccc(/C=C/c2ccc(Br)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.42
CA1 P00915 4/20 0.42
CA9 Q16790 4/20 0.42
CHRNA7 P36544 1/20 0.42
KDM4E B2RXH2 3/20 0.42
HPGD P15428 2/20 0.42
CYP2C19 P33261 2/20 0.42
RAB9A P51151 2/20 0.42
ALDH1A1 P00352 2/20 0.42
TUBB4A P04350 1/20 0.41
TUBB P07437 1/20 0.41
TUBA3C P0DPH7 1/20 0.41
TUBA1B P68363 1/20 0.41
TUBA4A P68366 1/20 0.41
TUBB4B P68371 1/20 0.41
TUBB3 Q13509 1/20 0.41
TUBB2A Q13885 1/20 0.41
TUBB8 Q3ZCM7 1/20 0.41
TUBA3E Q6PEY2 1/20 0.41
TUBA1A Q71U36 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8647806 1.00 CA12 (0.42) CA12CA1CA9CHRNA7KDM4E
SCHEMBL7189378 0.93 CA12 (0.46) CA12CA1CA9KDM4EHPGD
SCHEMBL614621 0.89 PREP (0.47) CA12CA1CA9KDM4ERAB9A
SCHEMBL6770995 0.87 PREP (0.46) CA12CA1CA9KDM4ERAB9A
SCHEMBL9699570 0.86 TRPA1 (0.53) CA12CA1CA9CHRNA7KDM4E
SCHEMBL3394945 0.84 CHRNA7 (0.49) CA12CA1CA9CHRNA7ALDH1A1
SCHEMBL21356550 0.84 ESR1 (0.50) CA12CA1CA9KDM4ERAB9A
SCHEMBL2607317 0.83 PREP (0.51) CA12CA1CA9KDM4EHPGD
SCHEMBL9843163 0.82 CA12 (0.42) CA12CA1CA9KDM4EHPGD
SCHEMBL9843159 0.82 CA12 (0.42) CA12CA1CA9KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0596057-B1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS ZENECA LTD (GB) 1998-09-09 EP disclosed
EP-0596057-A1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS ZENECA LIMITED (GB) 1994-05-11 EP disclosed
WO-1993021183-A1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS ZENECA LIMITED (GB) 1993-10-28 WO disclosed