SCHEMBL8649181

SCHEMBL8649181

COc1ccc2c(c1)C(CCN)=C(c1ccccc1)C2

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 2/20 0.61
HTR2A P28223 2/20 0.44
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
GAA P10253 1/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42
CYP2C19 P33261 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MTNR1A P48039 1/20 0.42
MTNR1B P49286 1/20 0.42
ACHE P22303 2/20 0.42
MAOB P27338 2/20 0.42
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA4 P22748 1/20 0.40
CA6 P23280 1/20 0.40
TAAR1 Q96RJ0 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7786867 0.99 NQO2 (0.60) NQO2HTR2AKDM4EALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL7779882 0.80 NQO2 (0.61) NQO2HTR2AKDM4EALDH1A1CYP1A2
SCHEMBL7784300 0.77 NQO2 (1.00) NQO2MTNR1AMTNR1B
SCHEMBL27547177 0.76 NQO2 (0.60) NQO2KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL4419991 0.75 ESR1 (0.53) NQO2KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL4895916 0.67 METAP1 (0.61) HTR2AKDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL10394812 0.67 METAP1 (0.46) NQO2HTR2AMTNR1AMTNR1BACHE
SCHEMBL10394815 0.67 METAP1 (0.46) NQO2HTR2AMTNR1AMTNR1BACHE
SCHEMBL3287680 0.67 ALDH1A1 (0.56) HTR2AKDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL3849905 0.67 ESR1 (0.59) NQO2ACHEMAOBNPY5RESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848699-A1 BENZOCYCLOALKENE COMPOUNDS WITH MELATONINE RECEPTOR BINDING AFFINITY, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-06-24 EP disclosed
EP-0781271-A1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1997-07-02 EP disclosed
WO-1997005098-A1 BENZOCYCLOALKENE COMPOUNDS WITH MELATONINE RECEPTOR BINDING AFFINITY, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-02-13 WO disclosed
WO-1996008466-A1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-21 WO disclosed