SCHEMBL8650467

SCHEMBL8650467

CCc1cc(C=O)c(OCc2ccccc2)cc1OCCCCCC(C)(C)C#N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 4/20 0.52
PDCD1 Q15116 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
LTB4R Q15722 3/20 0.37
CCNB2 O95067 1/20 0.37
CDK1 P06493 1/20 0.37
CDK4 P11802 1/20 0.37
CCNB1 P14635 1/20 0.37
CCND1 P24385 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
LTB4R2 Q9NPC1 2/20 0.36
SGMS2 Q8NHU3 1/20 0.36
ERN1 O75460 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8651806 0.88 NR1H4 (0.54) NR1H4LTB4RLTB4R2SGMS2
SCHEMBL8650341 0.88 NR1H4 (0.54) NR1H4LTB4RLTB4R2SGMS2HTR1A
SCHEMBL8560737 0.87 NR1H4 (0.53) NR1H4LTB4RLTB4R2SGMS2
SCHEMBL8651831 0.87 NR1H4 (0.53) NR1H4LTB4RLTB4R2
SCHEMBL8653472 0.87 NR1H4 (0.53) NR1H4LTB4RLTB4R2HTR1AADRA1D
SCHEMBL8568257 0.86 NR1H4 (0.52) NR1H4LTB4RLTB4R2
SCHEMBL6759095 0.85 NR1H4 (0.52) NR1H4LTB4RLTB4R2SGMS2
SCHEMBL8654007 0.85 NR1H4 (0.52) NR1H4LTB4RLTB4R2SGMS2KMT2A
SCHEMBL6757622 0.84 NR1H4 (0.51) NR1H4PDCD1CD274LTB4RLTB4R2
SCHEMBL8650436 0.84 NR1H4 (0.40) NR1H4CCNB2CDK1CDK4CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0579412-B1 1,2,4-trioxygenated benzene derivatives useful as a leukotriene antagonists LILLY CO ELI (US) 1998-10-07 EP disclosed
US-5352690-A For asthma, allergies ELI LILLY AND COMPANY (US) 1994-10-04 US disclosed
EP-0579412-A1 1,2,4-trioxygenated benzene derivatives useful as a leukotriene antagonists ELI LILLY AND COMPANY (US) 1994-01-19 EP disclosed