SCHEMBL8650341

SCHEMBL8650341

CCOc1cc(CC)c(OCCCCCC(C)(C)C#N)cc1OCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 4/20 0.54
HTR1A P08908 2/20 0.42
ADRA1D P25100 2/20 0.42
ADRA1A P35348 2/20 0.42
ADRA1B P35368 2/20 0.42
KDM4E B2RXH2 2/20 0.41
LMNA P02545 1/20 0.41
LTB4R Q15722 5/20 0.40
LTB4R2 Q9NPC1 4/20 0.40
MRGPRX4 Q96LA9 1/20 0.40
ALDH1A1 P00352 2/20 0.39
SGMS2 Q8NHU3 1/20 0.38
MAPK1 P28482 2/20 0.37
NTSR1 P30989 2/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
PKM P14618 1/20 0.37
HPGD P15428 1/20 0.37
HTT P42858 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8651806 0.94 NR1H4 (0.54) NR1H4LTB4RLTB4R2ALDH1A1SGMS2
SCHEMBL8653472 0.93 NR1H4 (0.53) NR1H4HTR1AADRA1DADRA1AADRA1B
SCHEMBL8654007 0.91 NR1H4 (0.52) NR1H4LTB4RLTB4R2ALDH1A1SGMS2
SCHEMBL8655412 0.90 NR1H4 (0.51) NR1H4KDM4ELTB4RLTB4R2SGMS2
SCHEMBL8651831 0.88 NR1H4 (0.53) NR1H4LTB4RLTB4R2
SCHEMBL8560737 0.88 NR1H4 (0.53) NR1H4LMNALTB4RLTB4R2SGMS2
SCHEMBL8650467 0.88 NR1H4 (0.52) NR1H4HTR1AADRA1DADRA1AADRA1B
SCHEMBL8568257 0.88 NR1H4 (0.52) NR1H4LTB4RLTB4R2
SCHEMBL8653660 0.87 NR1H4 (0.49) NR1H4KDM4ELMNALTB4RLTB4R2
SCHEMBL6759095 0.87 NR1H4 (0.52) NR1H4LMNALTB4RLTB4R2SGMS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0579412-B1 1,2,4-trioxygenated benzene derivatives useful as a leukotriene antagonists LILLY CO ELI (US) 1998-10-07 EP disclosed
US-5352690-A For asthma, allergies ELI LILLY AND COMPANY (US) 1994-10-04 US disclosed
EP-0579412-A1 1,2,4-trioxygenated benzene derivatives useful as a leukotriene antagonists ELI LILLY AND COMPANY (US) 1994-01-19 EP disclosed