SCHEMBL8650900

SCHEMBL8650900

Cc1ccc(/C(=C\c2ccccc2Cl)C(=O)NC(=N)N)cn1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.39
RAB9A P51151 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
NPC1 O15118 2/20 0.39
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
ALDH1A1 P00352 3/20 0.37
LMNA P02545 2/20 0.37
MAPT P10636 2/20 0.36
NPSR1 Q6W5P4 3/20 0.36
ADORA3 P0DMS8 1/20 0.36
MEN1 O00255 2/20 0.35
HPGD P15428 1/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 2/20 0.35
ATM Q13315 1/20 0.35
KLF5 Q13887 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8643112 0.96 KMT2A (0.37) KMT2ARAB9ASMN1; SMN2NPC1HDAC1
SCHEMBL8643120 0.84 MAPT (0.51) KMT2ARAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL8643116 0.84 KMT2A (0.37) KMT2ARAB9ASMN1; SMN2NPC1HDAC1
SCHEMBL8646247 0.82 MAPT (0.46) KMT2ARAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL8644175 0.81 KMT2A (0.43) KMT2ARAB9ASMN1; SMN2NPC1HDAC1
SCHEMBL8644173 0.81 KMT2A (0.43) KMT2ARAB9ASMN1; SMN2NPC1HDAC1
SCHEMBL8646364 0.76 MAPT (0.44) KMT2ARAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL8649037 0.75 ATM (0.42) KMT2ARAB9ASMN1; SMN2NPC1HDAC1
SCHEMBL19341349 0.74 CA1 (0.43) KMT2ARAB9ASMN1; SMN2NPC1HDAC1
SCHEMBL8648196 0.72 HDAC1 (0.46) KMT2ARAB9ANPC1HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861831-A1 HETEROARYL-SUBSTITUTED ACRYLOYLGUANIDINE DERIVATIVES AND MEDICINAL COMPOSITION THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-09-02 EP disclosed