SCHEMBL8655705

SCHEMBL8655705

O=CCCC[C@@H](C(=O)OCc1ccccc1)N1C(=O)c2ccccc2C1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.51
ALDH1A1 P00352 5/20 0.49
GAA P10253 1/20 0.49
POLB P06746 3/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
HSD11B1 P28845 1/20 0.46
MAPK1 P28482 2/20 0.45
KDM4E B2RXH2 1/20 0.45
TP53 P04637 1/20 0.45
GLA P06280 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
HPGD P15428 1/20 0.45
ALOX12 P18054 1/20 0.45
NFKB1 P19838 1/20 0.45
APEX1 P27695 1/20 0.45
HSD17B10 Q99714 1/20 0.45
PKM P14618 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8655711 1.00 HTT (0.51) HTTALDH1A1GAAPOLBL3MBTL1
SCHEMBL11057185 0.85 HTT (0.53) HTTALDH1A1GAAPOLBL3MBTL1
SCHEMBL10725924 0.85 HTT (0.53) HTTALDH1A1GAAPOLBL3MBTL1
SCHEMBL10725915 0.85 HTT (0.53) HTTALDH1A1GAAPOLBL3MBTL1
SCHEMBL30278688 0.84 ALDH1A1 (0.46) HTTALDH1A1GAAPOLBHSD11B1
SCHEMBL21895832 0.84 ALDH1A1 (0.46) HTTALDH1A1GAAPOLBHSD11B1
SCHEMBL21895831 0.84 ALDH1A1 (0.46) HTTALDH1A1GAAPOLBHSD11B1
SCHEMBL7349201 0.83 ALDH1A1 (0.64) ALDH1A1GAAPOLBL3MBTL1MAPK1
SCHEMBL7349189 0.83 ALDH1A1 (0.64) ALDH1A1GAAPOLBL3MBTL1MAPK1
SCHEMBL10166837 0.81 ALDH1A1 (0.42) HTTALDH1A1GAAPOLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5723602-A ANGIOTENSIN CONVERTING ENZYME AND ENDOPEPTIDASE INHIBITORS, CARDIOVASCULAR DISORDERS E. R. SQUIBB & SONS, INC. (US) 1998-03-03 US disclosed
US-4661479-A ENZYME INHIBITORS MERCK AND CO., INC. (US) 1987-04-28 US disclosed
EP-0061187-B1 BICYCLIC LACTAMS AS ANTIHYPERTENSIVES MERCK & CO. INC. (US) 1986-08-20 EP disclosed
US-4415496-A HYPOTENSIVE AGENTS; 5-OXOTHIAZOLO/3,2-A/AZEPINE DERIVATIVES FROM A PHTHALIMIDE MERCK & CO., INC. (US) 1983-11-15 US disclosed
EP-0061187-A1 Bicyclic lactams as antihypertensives MERCK & CO. INC. (US) 1982-09-29 EP disclosed