SCHEMBL8656362

SCHEMBL8656362

O=C(O)/C=C1/CCc2cc3ccccc3n2C1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.42
HTR2C P28335 5/20 0.42
NOTUM Q6P988 1/20 0.42
SIGMAR1 Q99720 12/20 0.39
DAO P14920 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21028290 0.81 HTR2A (0.42) HTR2AHTR2CSIGMAR1
SCHEMBL235219 0.73 NOTUM (0.59) HTR2AHTR2CNOTUMSIGMAR1
SCHEMBL19930594 0.73 HTR2A (0.53) HTR2AHTR2CNOTUMSIGMAR1
SCHEMBL20080086 0.70 HTR2A (0.50) HTR2AHTR2CNOTUMSIGMAR1
SCHEMBL8447696 0.70 HTR2A (0.43) HTR2AHTR2CNOTUMSIGMAR1DAO
Acetic Acid SCHEMBL13279290 0.68 HTR2A (0.55) HTR2AHTR2CSIGMAR1
SCHEMBL13279281 0.67 HTR2A (0.40) HTR2AHTR2CNOTUMSIGMAR1DAO
SCHEMBL8449826 0.66 MAPT (0.42) HTR2AHTR2CNOTUMSIGMAR1DAO
SCHEMBL10735669 0.66 HTR2A (0.56) HTR2AHTR2CNOTUMSIGMAR1
SCHEMBL30684257 0.66 HTR2A (0.56) HTR2AHTR2CNOTUMSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721245-A ANTIINFLAMMATORY AGENTS, RESPIRATORY SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS HOFFMANN-LA ROCHE INC. (US) 1998-02-24 US disclosed
EP-0384349-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1994-04-27 EP disclosed
EP-0384349-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1990-08-29 EP disclosed