SCHEMBL8447696

SCHEMBL8447696

O=C(O)C1CCc2cc3ccccc3n2C1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.43
HTR2C P28335 5/20 0.43
NOTUM Q6P988 4/20 0.42
SIGMAR1 Q99720 4/20 0.41
AKR1C3 P42330 5/20 0.41
AKR1C1 Q04828 2/20 0.41
DAO P14920 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8447283 0.87 HTR2A (0.49) HTR2AHTR2CNOTUMSIGMAR1AKR1C3
SCHEMBL8449826 0.85 MAPT (0.42) HTR2AHTR2CNOTUMSIGMAR1AKR1C3
SCHEMBL8450915 0.83 HTR2A (0.43) HTR2AHTR2CSIGMAR1
SCHEMBL21027979 0.83 HTR2A (0.43) HTR2AHTR2CSIGMAR1
SCHEMBL8328343 0.80 ALDH1A1 (0.45) HTR2AHTR2C
SCHEMBL8450784 0.79 HTR2A (0.39) HTR2AHTR2CSIGMAR1
SCHEMBL13279281 0.79 HTR2A (0.40) HTR2AHTR2CNOTUMSIGMAR1DAO
SCHEMBL233436 0.78 HTR2A (0.47) HTR2AHTR2CNOTUMSIGMAR1
SCHEMBL8452782 0.77 HTR2A (0.44) HTR2AHTR2CNOTUMSIGMAR1AKR1C3
SCHEMBL8454162 0.77 HTR2A (0.44) HTR2AHTR2CNOTUMSIGMAR1AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0624586-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-09-01 EP disclosed
US-5721230-A ANTIINFLAMMATORY AGENT, VIRICIDES; TREATING CARDIOVASCULAR DISORDER, RESPIRATORY SYSTEM DISORDER, THROMBOSIS, DIABETES, ALOPECIA HOFFMANN-LA ROCHE INC. (US) 1998-02-24 US disclosed
EP-0624586-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1994-11-17 EP disclosed