SCHEMBL8657665

SCHEMBL8657665

Cc1ccc(Oc2c(C)cc(NC(=O)NC(=O)c3ccccc3Cl)c(C)c2Cl)c(Br)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYGL P06737 6/20 0.49
RAB9A P51151 2/20 0.44
GCGR P47871 1/20 0.43
KMT2A Q03164 3/20 0.43
GAA P10253 2/20 0.43
MAPT P10636 2/20 0.43
ALDH1A1 P00352 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41
PKM P14618 1/20 0.41
MEN1 O00255 2/20 0.41
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
IDO1 P14902 1/20 0.38
TP53 P04637 1/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9135160 0.93 PYGL (0.49) PYGLRAB9AGCGRKMT2AALDH1A1
SCHEMBL8663054 0.93 PYGL (0.49) PYGLRAB9AGCGRGAAMAPT
SCHEMBL8658014 0.91 PYGL (0.52) PYGLRAB9AGCGRKMT2AGAA
SCHEMBL8657590 0.91 PYGL (0.49) PYGLRAB9AGCGRKMT2AGAA
SCHEMBL10492145 0.90 PYGL (0.51) PYGLRAB9AGCGRKMT2AGAA
SCHEMBL8660846 0.90 PYGL (0.48) PYGLRAB9AGCGRKMT2AGAA
SCHEMBL8661667 0.89 PYGL (0.49) PYGLRAB9AGCGRKMT2AGAA
SCHEMBL8658946 0.88 PYGL (0.50) PYGLRAB9AGCGRGAAMAPT
SCHEMBL9137528 0.86 PYGL (0.53) PYGLRAB9AGCGRKMT2AGAA
SCHEMBL8656634 0.86 PYGL (0.52) PYGLRAB9AGCGRKMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
US-4873264-A Novel pesticidal 1-(alkyl-phenoxy-aryl)-3-benzoyl ureas and process for preparation RHONE-POULENC NEDERLANDS B.V. (NL) 1989-10-10 US disclosed
EP-0098158-B1 PESTICIDAL 1-(ALKYL-PHENOXYARYL)-3-BENZOYL UREAS AND PROCESS FOR PREPARATION UNION CARBIDE CORPORATION (US) 1987-11-19 EP disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed
EP-0124283-A1 Process for the preparation of benzoyl ureas UNION CARBIDE CORPORATION (US) 1984-11-07 EP disclosed
EP-0098158-A1 Pesticidal 1-(alkyl-phenoxyaryl)-3-benzoyl ureas and process for preparation UNION CARBIDE CORPORATION (US) 1984-01-11 EP disclosed