P-Xylene

P-Xylene

SCHEMBL8660591

Cc1ccc(C)cc1.Cc1ccc(S(=O)(=O)O)cc1

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1BMXBRAFBTKCHRNA4CHRNB2CSNK1EEGFRERBB2F10FLT1FLT3FLT4IGF1RINSRITKJAK3KDRKITOPRM1PARP1PARP2PDGFRBPIK3CDRAF1RETSLC18A2TECTXKdacAdacBdacCftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of P-Xylene. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.62
LMNA P02545 2/20 0.59
ALDH1A1 P00352 5/20 0.58
SMN1; SMN2 Q16637 3/20 0.58
TDP1 Q9NUW8 2/20 0.58
KDM4E B2RXH2 1/20 0.58
MAPT P10636 1/20 0.58
HTT P42858 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
CA1 P00915 2/20 0.56
CA2 P00918 2/20 0.56
TSHR P16473 2/20 0.56
CA12 O43570 1/20 0.56
CA3 P07451 1/20 0.56
CA6 P23280 1/20 0.56
CA5A P35218 1/20 0.56
CA7 P43166 1/20 0.56
CA9 Q16790 1/20 0.56
CA5B Q9Y2D0 1/20 0.56
NT5E P21589 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29991938 1.00 GAA (0.62) GAALMNAALDH1A1SMN1; SMN2TDP1
SCHEMBL34 1.00 GAA (0.62) GAALMNAALDH1A1SMN1; SMN2TDP1
SCHEMBL5068661 1.00 GAA (0.62) GAALMNAALDH1A1SMN1; SMN2TDP1
SCHEMBL31313 1.00 GAA (0.62) GAALMNAALDH1A1SMN1; SMN2TDP1
SCHEMBL11432043 1.00 GAA (0.62) GAALMNAALDH1A1SMN1; SMN2TDP1
SCHEMBL1705904 1.00 GAA (0.62) GAALMNAALDH1A1SMN1; SMN2TDP1
SCHEMBL1594407 0.97 GAA (0.59) GAALMNAALDH1A1SMN1; SMN2TDP1
Water SCHEMBL214962 0.97 GAA (0.59) GAALMNAALDH1A1SMN1; SMN2TDP1
SCHEMBL1345322 0.97 GAA (0.59) GAALMNAALDH1A1SMN1; SMN2TDP1
SCHEMBL22802539 0.97 GAA (0.59) GAALMNAALDH1A1SMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0242620-B1 MODIFIED PHENOLIC FOAM CATALYSTS AND METHOD FIBERGLAS CANADA Inc. (CA) 1991-06-12 EP claimed
US-4945077-A Aromatic sulfonic acid and resorcinol FIBERGLASS CANADA INC. (CA) 1990-07-31 US claimed
US-4883824-A AROMATIC SULFONIC ACID AND DIHYDRIC PHENOL TO PRODUCE CLOSED CELL FOAM FIBERGLAS CANADA, INC. (CA) 1989-11-28 US claimed
US-5786398-A PHENOL-FORMALDEHYDE RESINS; THERMOCONDUCTIVITY OWENS-CORNING FIBERGLAS TECHNOLOGY INC. (US) 1998-07-28 US disclosed
EP-0815163-A1 INSULATING FOAMS AND THE MANUFACTURING THEREOF OWENS CORNING (US) 1998-01-07 EP disclosed
EP-0579321-B1 Process for producing a mainly closed cell phenolic foam RECTICEL (BE) 1997-09-03 EP disclosed
WO-1996030437-A1 INSULATING FOAMS AND THE MANUFACTURING THEREOF OWENS CORNING (US) 1996-10-03 WO disclosed
EP-0579321-A1 Process for producing a mainly closed cell phenolic foam RECTICEL (BE) 1994-01-19 EP disclosed
EP-0242620-B1 MODIFIED PHENOLIC FOAM CATALYSTS AND METHOD FIBERGLAS CANADA Inc. (CA) 1991-06-12 EP disclosed
US-4945077-A Aromatic sulfonic acid and resorcinol FIBERGLASS CANADA INC. (CA) 1990-07-31 US disclosed
US-4883824-A AROMATIC SULFONIC ACID AND DIHYDRIC PHENOL TO PRODUCE CLOSED CELL FOAM FIBERGLAS CANADA, INC. (CA) 1989-11-28 US disclosed
EP-0242620-A2 Modified phenolic foam catalysts and method FIBERGLAS CANADA Inc. (CA) 1987-10-28 EP disclosed