SCHEMBL8660848

SCHEMBL8660848

Cc1cc(Oc2cc(Cl)c(Cl)cc2Br)c(Cl)c(C)c1NC(=O)NC(=O)c1c(F)cccc1Cl

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MAPT P10636 4/20 0.40
POLB P06746 2/20 0.40
USP2 O75604 1/20 0.40
ALOX15 P16050 1/20 0.40
GAA P10253 5/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAPK1 P28482 2/20 0.39
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PPIA P62937 1/20 0.39
ATM Q13315 1/20 0.38
PKM P14618 1/20 0.38
TLR8 Q9NR97 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27694017 0.93 MAPT (0.43) MEN1KMT2AMAPTPOLBMAPK1
SCHEMBL8660856 0.92 MEN1 (0.45) MEN1KMT2AMAPTPOLBUSP2
SCHEMBL8663050 0.91 MEN1 (0.41) MEN1KMT2AMAPTPOLBUSP2
SCHEMBL8658883 0.91 MEN1 (0.41) MEN1KMT2AMAPTPOLBUSP2
SCHEMBL8660912 0.89 KMT2A (0.43) MEN1KMT2AMAPTGAAL3MBTL1
SCHEMBL8659947 0.88 KMT2A (0.48) MEN1KMT2AMAPTPOLBUSP2
SCHEMBL8658546 0.86 MEN1 (0.43) MEN1KMT2AMAPTPOLBUSP2
SCHEMBL8660739 0.86 MEN1 (0.43) MEN1KMT2AMAPTPOLBUSP2
SCHEMBL8660959 0.85 PYGL (0.47) MEN1KMT2AMAPTPOLBL3MBTL1
SCHEMBL9138753 0.85 MEN1 (0.39) MEN1KMT2AMAPTPOLBUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed