SCHEMBL8661978

SCHEMBL8661978

CCCC(=O)Oc1ccc(C#Cc2ccc3c(c2)C(CC)(CC)CCS3)s1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.40
RARA P10276 2/20 0.40
RARB P10826 2/20 0.40
RARG P13631 2/20 0.40
KMT2A Q03164 1/20 0.40
CYP26A1 O43174 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7817653 0.89 RARA (0.42) CYP3A4RARARARBRARGKMT2A
SCHEMBL8659637 0.86
SCHEMBL8664820 0.85
SCHEMBL8664182 0.82 CYP3A4 (0.47) CYP3A4RARARARBRARGKMT2A
SCHEMBL8660133 0.82
SCHEMBL8659480 0.80 CYP3A4 (0.40) CYP3A4RARARARBRARGKMT2A
SCHEMBL8662237 0.80 CYP3A4 (0.47) CYP3A4RARARARBRARGKMT2A
SCHEMBL8661983 0.79 CYP3A4 (0.46) CYP3A4RARARARBRARGKMT2A
SCHEMBL8662227 0.79 CYP3A4 (0.50) CYP3A4RARARARBRARGKMT2A
SCHEMBL7651204 0.79 RARA (0.41) CYP3A4RARARARBRARGKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750693-A THIOCHROMANYL OR CHROMANYL COMPOUNDS AS ANTICARCINOGINIC AGENTS, SKIN DISORDERS AND ATHEROSCLEROSIS ALLERGAN (US) 1998-05-12 US disclosed
US-5677451-A CONTROLLING CELL DIFFERENTIATION; SKIN DISORDERS; ANTICANCER AGENTS ALLERGAN (US) 1997-10-14 US disclosed