SCHEMBL8663003

SCHEMBL8663003

COc1cc(-c2ccccc2-c2ccccc2S(N)(=O)=O)cc(OC)c1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.51
PTGS1 P23219 3/20 0.51
PTGES2 Q9H7Z7 4/20 0.43
CA12 O43570 3/20 0.41
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
CA9 Q16790 3/20 0.41
BRD4 O60885 1/20 0.41
PKM P14618 2/20 0.40
SCN9A Q15858 1/20 0.39
ERN1 O75460 1/20 0.39
PTPRC P08575 1/20 0.39
PTPN1 P18031 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
DUSP3 P51452 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8657816 0.88 PTGS2 (0.50) PTGS2PTGS1PTGES2ERN1
SCHEMBL8661248 0.87 PTGS2 (0.46) PTGS2PTGS1PTGES2CA12CA1
SCHEMBL8656781 0.87 CA9 (0.54) PTGS2PTGS1CA12CA1CA2
SCHEMBL8659792 0.86 PTGS2 (0.59) PTGS2PTGS1PTGES2CA12CA1
SCHEMBL8659436 0.86 PTGS2 (0.51) PTGS2PTGS1CA12CA1CA2
SCHEMBL8661261 0.84 PTGS1 (0.40) PTGS2PTGS1PTGES2CA12CA1
SCHEMBL8660023 0.83 PTGS2 (0.74) PTGS2PTGS1PTGES2BRD4PTPRC
SCHEMBL6733291 0.83 PTGS2 (0.73) PTGS2PTGS1CA12CA1CA2
SCHEMBL8656732 0.83 PTGS2 (0.53) PTGS2PTGS1PTGES2CA1CA2
SCHEMBL8657870 0.82 PTGS2 (0.45) PTGS2PTGS1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739166-A ALKYLSULFONYL OR AMINOSULFONYL SUBSTITUTED AROMATIC COMPOUNDS AS NON-STEROIDAL ANTIINFLAMMATORY AGENT G.D. SEARLE & CO. (US) 1998-04-14 US disclosed