SCHEMBL8663176

SCHEMBL8663176

Cc1cc(NC(=O)NC(=O)c2c(Cl)cccc2Cl)c(C)c(Cl)c1Oc1ccc(Cl)cc1Br

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.39
MAPT P10636 3/20 0.39
POLB P06746 2/20 0.39
PYGL P06737 6/20 0.38
PARP1 P09874 1/20 0.38
PARG Q86W56 1/20 0.38
CXCR2 P25025 1/20 0.37
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
GCGR P47871 1/20 0.36
GHSR Q92847 1/20 0.36
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
ALOX12 P18054 1/20 0.35
ATM Q13315 1/20 0.35
ALDH1A1 P00352 2/20 0.35
THRB P10828 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8660941 0.94 MEN1 (0.45) NPSR1MAPTPOLBKMT2AMEN1
SCHEMBL8660569 0.92 POLB (0.39) MAPTPOLBPYGLKMT2AMEN1
SCHEMBL8657546 0.91 NPSR1 (0.45) NPSR1MAPTPYGLKMT2AMEN1
SCHEMBL8661612 0.91 NPSR1 (0.42) NPSR1MAPTPOLBPYGLPARP1
SCHEMBL8659309 0.91 MEN1 (0.47) NPSR1MAPTPOLBPYGLPARP1
SCHEMBL9135160 0.90 PYGL (0.49) POLBPYGLPARP1PARGCXCR2
SCHEMBL8660863 0.89 POLB (0.38) MAPTPOLBPYGLKMT2AMEN1
SCHEMBL10762785 0.87 MAPT (0.38) NPSR1MAPTPOLBPYGLPARP1
SCHEMBL8656921 0.87 KMT2A (0.38) NPSR1MAPTPOLBPYGLPARP1
SCHEMBL8659821 0.86 MEN1 (0.45) NPSR1MAPTPOLBKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed