Indole

Indole

SCHEMBL8664418

C=O.NCC(=O)O.c1ccc2[nH]ccc2c1

nearest known ligand 0.59

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Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3PDE3APDE3BPDE4APDE4BPDE4CPDE4D

The experimentally established mechanism targets of Indole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.59
CA1 P00915 1/20 0.59
CA2 P00918 1/20 0.59
ITGB2 P05107 1/20 0.59
ICAM1 P05362 1/20 0.59
ITGAL P20701 1/20 0.59
CA4 P22748 1/20 0.59
CA6 P23280 1/20 0.59
AHR P35869 1/20 0.59
ADK P55263 1/20 0.59
CTNNB1 P35222 1/20 0.45
WNT3A P56704 1/20 0.45
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
ENPP2 Q13822 2/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
NPC1 O15118 2/20 0.41
MAPT P10636 2/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Indole SCHEMBL16757645 0.96 TRPA1 (0.63) TRPA1CA1CA2ITGB2ICAM1
Indole SCHEMBL28576095 0.95 TRPA1 (0.61) TRPA1CA1CA2ITGB2ICAM1
Indole SCHEMBL28967497 0.92 TRPA1 (0.57) TRPA1CA1CA2ITGB2ICAM1
Indole SCHEMBL2170920 0.86 TRPA1 (0.59) TRPA1CA1CA2ITGB2ICAM1
Indole SCHEMBL6925060 0.86 TRPA1 (0.63) TRPA1CA1CA2ITGB2ICAM1
Indole SCHEMBL6835663 0.84 TRPA1 (0.65) TRPA1CA1CA2ITGB2ICAM1
Indole SCHEMBL1714414 0.84 TRPA1 (0.65) TRPA1CA1CA2ITGB2ICAM1
Indole SCHEMBL384964 0.83 TRPA1 (0.71) TRPA1CA1CA2ITGB2ICAM1
Indole SCHEMBL28479409 0.83 TRPA1 (0.77) TRPA1CA1CA2ITGB2ICAM1
Indole SCHEMBL5851080 0.83 AHR (0.85) TRPA1CA1CA2ITGB2ICAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776740-A Process for the preparation of L-tryptophan MITSUBISHI CHEMICAL CORPORATION (JP) 1998-07-07 US disclosed