SCHEMBL8664434

SCHEMBL8664434

O[N][C@H]1CCc2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.46
PDPK1 O15530 1/20 0.46
CYP11B2 P19099 1/20 0.43
ACP3 P15309 1/20 0.41
PIN1 Q13526 1/20 0.41
ADRA1A P35348 1/20 0.41
SLC18A3 Q16572 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
RET P07949 1/20 0.39
HTR2A P28223 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4185301 1.00 IDO1 (0.46) IDO1PDPK1CYP11B2ACP3PIN1
SCHEMBL2322453 0.83 IDO1 (0.48) IDO1PDPK1CYP11B2CA1CA2
SCHEMBL29980773 0.83 IDO1 (0.48) IDO1PDPK1CYP11B2CA1CA2
SCHEMBL5085348 0.79 PDPK1 (0.50) IDO1PDPK1CYP11B2ADRA1A
SCHEMBL20321008 0.79 IDO1 (0.46) IDO1PDPK1CYP11B2CA1CA2
SCHEMBL2400656 0.79 PDPK1 (0.50) IDO1PDPK1CYP11B2ADRA1A
SCHEMBL1148775 0.75 IDO1 (0.42) IDO1PDPK1CYP11B2PIN1ADRA1A
SCHEMBL2541173 0.75 IDO1 (0.42) IDO1PDPK1CYP11B2ADRA1ACA1
SCHEMBL13435342 0.75 IDO1 (0.42) IDO1PDPK1CYP11B2ACP3
SCHEMBL1922245 0.75 IDO1 (0.42) IDO1PDPK1CYP11B2ADRA1ACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0601486-B1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD (KR) 1997-10-29 EP claimed
EP-0601486-A1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD. (KR) 1994-06-15 EP claimed
US-5763631-A CIS-EPOXIDE COMPOUNDS; ANTIVIRUS AGENTS; USEFUL TO TREAT THE AIDS LUCKY LIMITED (KR) 1998-06-09 US disclosed
US-5744621-A CIS-EPOXIDE COMPOUNDS LUCKY LIMITED. (KR) 1998-04-28 US disclosed
EP-0601486-B1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD (KR) 1997-10-29 EP disclosed
US-5587388-A AIDS; VIRICIDES LUCKY LIMITED (KR) 1996-12-24 US disclosed
EP-0601486-A1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD. (KR) 1994-06-15 EP disclosed