SCHEMBL8664436

SCHEMBL8664436

ON[C@H]1CCc2ccccc21

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.66
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
SLC18A3 Q16572 1/20 0.56
MAOA P21397 4/20 0.54
MAOB P27338 4/20 0.54
BCHE P06276 1/20 0.54
ADRA2B P18089 1/20 0.54
ADRA2C P18825 1/20 0.54
ACHE P22303 1/20 0.54
ADRA1A P35348 1/20 0.54
HTR6 P50406 1/20 0.54
KDM1A O60341 1/20 0.51
FADS1 O60427 1/20 0.50
TAS1R3 Q7RTX0 1/20 0.47
TAS1R1 Q7RTX1 1/20 0.47
TAS1R2 Q8TE23 1/20 0.47
HTT P42858 1/20 0.46
EPHX2 P34913 2/20 0.46
IDO1 P14902 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2321988 1.00 PDPK1 (0.66) PDPK1CA1CA2SLC18A3MAOA
SCHEMBL6344102 0.88 HTT (0.59) TAS1R3TAS1R1TAS1R2HTTALDH1A1
SCHEMBL2322457 0.83 PDPK1 (0.70) PDPK1CA1CA2SLC18A3MAOA
Hydrochloric Acid SCHEMBL7123292 0.81 PDPK1 (0.68) PDPK1CA1CA2SLC18A3MAOA
SCHEMBL19508305 0.79 PDPK1 (0.66) PDPK1CA1CA2SLC18A3MAOA
SCHEMBL20354303 0.79 PDPK1 (0.66) PDPK1CA1CA2SLC18A3MAOA
SCHEMBL61508 0.79 PDPK1 (1.00) PDPK1CA1CA2SLC18A3MAOA
SCHEMBL1488037 0.79 PDPK1 (0.66) PDPK1CA1CA2SLC18A3MAOA
SCHEMBL6850366 0.79 PDPK1 (0.66) PDPK1CA1CA2SLC18A3MAOA
SCHEMBL13618841 0.79 PDPK1 (0.66) PDPK1CA1CA2SLC18A3MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0601486-B1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD (KR) 1997-10-29 EP claimed
EP-0601486-A1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD. (KR) 1994-06-15 EP claimed
CN-1222909-A Pyrazinone thrombin inhibitors MERCK & CO INC (US) 1999-07-14 CN disclosed
US-5763631-A CIS-EPOXIDE COMPOUNDS; ANTIVIRUS AGENTS; USEFUL TO TREAT THE AIDS LUCKY LIMITED (KR) 1998-06-09 US disclosed
US-5744621-A CIS-EPOXIDE COMPOUNDS LUCKY LIMITED. (KR) 1998-04-28 US disclosed
EP-0601486-B1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD (KR) 1997-10-29 EP disclosed
US-5587388-A AIDS; VIRICIDES LUCKY LIMITED (KR) 1996-12-24 US disclosed
EP-0601486-A1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD. (KR) 1994-06-15 EP disclosed